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publicationDate 2014-07-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2011256444-B2
titleOfInvention Spiro isoxazoline compounds as SSTR5 antagonists
abstract Substituted spirocyclic amines of structural formula (I) are selective antagonists of the somatostatin subtype receptor 5 (SSTR5) and are useful for the treatment, control or prevention of disorders responsive to antagonism of SSTR5, such as Type 2 diabetes, insulin resistance, lipid disorders, obesity, atherosclerosis, Metabolic Syndrome, depression, and anxiety.
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Total number of triples: 1807.