http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AU-2010236027-B2

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filingDate 2010-10-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2011-08-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3c028b69acb681fafde56de11b7c5c70
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publicationDate 2011-08-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2010236027-B2
titleOfInvention 2-pyrazinone derivatives for the treatment of disease or condition in which inhibition of neutrophil elastase activity is beneficial
abstract NOVEL COMPOUNDS II 5 The invention provides compounds of formula R 14 W N N X-R 5 (1) wherein R , R3, R4, R , R , X and W are as defined in the specification and optical isomers, racemates and tautomers thereof, and pharmaceutically acceptable salts thereof, 10 together with processes for their preparation, pharmaceutical compositions containing them and their use in therapy. The compounds are inhibitors of human neutrophil elastase.
priorityDate 2006-05-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419494150
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4L800
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54585
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393749
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID713
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100328627
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ97F65
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403802
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3565
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419532830
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0K1F4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID14517
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504776
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281161
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1253269
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13157
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ97R22
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419501187
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP25524
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1234
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281160
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID107735
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID17392
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97513
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP13109
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152743293
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7CXF9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9294
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ865X5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419569347
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419505994
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID17386
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25317
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458394763
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5QWC7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454031468
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5MBA8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3652
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID17385
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID607724
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415748971
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456468049
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID57133995
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID46937068
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534234
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506983
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3052776
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5NH50
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID282871
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54385
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9973510
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97398
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5339

Total number of triples: 1329.