http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AU-2010218853-A1

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inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_763ba6b59f6f290fb3a4d9c88305c2f5
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publicationDate 2011-10-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2010218853-A1
titleOfInvention Tricyclic pyrazolopyrimidine derivative
abstract Disclosed is a novel compound which inhibits an activity of HSP90, in particular a novel compound which inhibits a function of HSP90 as a chaperone protein and has an antitumor activity. Specifically disclosed are: a pyrazolopyrimidine compound represented by formula (1) having various substituents, which inhibits an ATPase activity of HSP90 and has an antitumor activity; an HSP90 inhibitor which contains a compound represented by formula (1); a pharmaceutical formulation which contains a compound represented by formula (1); an antitumor agent which contains a compound represented by formula (1); a pharmaceutical composition which contains a compound represented by formula (1); and a method for treating a cancer, wherein a compound represented by formula (1) is used.
priorityDate 2009-02-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 446.