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filingDate 2008-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-02-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f8b72e6d8d2f8a8c4861c291cff0e6b4
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publicationDate 2015-02-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2008268262-C1
titleOfInvention MetAP-2 inhibitor polymersomes for therapeutic administration
abstract Described herein are MetAP-2 inhibitors and compositions and formulations thereof, and more particularly compositions and formulations of MetAP-2 inhibitors wherein the MetAP-2 inhibitor is associated with a block copolymer comprising a hydrophilic polymer moiety and a hydrophobic polymer moiety. The present invention also relates to compositions and formulations comprising MetAP-2 inhibitors for oral administration or administration via routes such as topical or ocular administration. The present invention also provides methods to treat conditions associated with or related to the over-expression or over-activity of MetAP-2 by administering the compositions and formulations comprising MetAP-2 inhibitors as disclosed herein.
priorityDate 2007-06-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426079160
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP20003
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411212574
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID83785
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID676246
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DQH9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4RDI6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554352
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426343843
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419479687
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450311443
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8SR45
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419580923
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO19002
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP09038
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID396495
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60791
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7953
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492167
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID174260
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID77991
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ59LF9
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID72172
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WK19
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP16612
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7YRB5
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP9WK18
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8617632
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID56307
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403727
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID28417
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP19874
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID513497
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID641462
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23543135
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281161
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD1ZEN1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414100136
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID84310
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44357137
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5394
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID83783
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4YSA9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10631
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID10988
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID30487
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08317
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP50412
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP03969
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7EZ86
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419536599
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID374100
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID407170
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3001055
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID99824
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419590905
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD4DE65
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53865415
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4Y1F8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100101279
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9427
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCD4B2G3
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5P8Q4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID430778997
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280828
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5M8M4
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419874183
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID482154
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCX2JCV5
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2092
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID14254
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3ZC89
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4R2P3
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3152
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP15692
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID222778
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2724247
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9829523
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID65163
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Total number of triples: 466.