http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AU-2008201395-B2

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filingDate 2008-03-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-08-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3107124f61dac6d869b1662d680a7faa
publicationDate 2013-08-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2008201395-B2
titleOfInvention Short term sustained drug-delivery system for implantable medical devices and method of making the same
abstract A short-term sustained drug eluting coating for implantable medical devices is disclosed. The coating comprises a biocompatible matrix and at least one pharmacologically or biologically active agent and releases substantially one of all of 5 its payloads within four to six weeks post-implantation. When a combination of pharmacological agents are incorporated in the disclosed sustained drug eluting matrix of a drug/device combination, at least one agent is preferred to substantially release in a short duration. Medical devices benefiting from such a desired sustained drug eluting coating include drug eluting cardiovascular, peripheral, and 10 neurovascular stents, abdominal aortic aneurysm (AAA) prosthesis, anastomosis shunt, arterial/venous (AV) shunts etc. One embodiment of the invention is a sustained release coating or depot on or in a stent that releases substantially all of it payload for ischemic myocardial injury after a heart attack. The coating may be formed from biocompatible stable and absorbable polymers of natural and synthetic 15 origins. Useful pharmacological agents for inhibiting vascular neointimal growth post-angioplasty that leads to restenosis include macrolide polyenes such as a rapamycin and all its derivatives and analogs; paclitaxel and all derivatives and analogs. Useful agents for other vascular conditions such as vulnerable plaques may comprise anti-inflammatory, anti-proliferative agents, and matrix metalloprotease 20 (MMP) inhibitors. 26/03/08,kn 17213 spcification,30 14 0- 18C 23c 20 2 .- 30 o o O 230b
priorityDate 2007-03-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60947
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426079013
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67971
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419583338
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP41522
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407139333
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67974
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27007
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9MYV3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67968
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP96471
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67965
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DJG0
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID296456
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67969
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502152
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF7HUS6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ00731
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF7FQM7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6JV22
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480215
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DJG1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426149262
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504459
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID454269980
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID409982724
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0K3N5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID25244225
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423217529
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCH0VVW3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4211
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP33708
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID222786
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP48617
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP33707
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCG5BQH5
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419590872
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419491660
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0K3N4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07321
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419533737
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2754
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2056
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCG3QY98
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100151255
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9942124
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP02648
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422601179
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4NWI1
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5554
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5282448
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2123
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9NDE7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID463609
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281408
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5555
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4QHB1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4GGF2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419505112
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID227
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419590725
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4JVW6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419552660
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68245
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534036
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502143
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB4HT15
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID36314
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281407
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419480574
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68243
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415968435
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419534242
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31307
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GKR0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9GKA2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9782
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ21697
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60606
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8MR45
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100002479
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP42633
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4T554
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ867B1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426222649
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419552610
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415713612
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9W7R2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504692
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419506265
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8MHY7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP29598
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415970532
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4R6C4
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403802
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID479427
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCH0ZG98
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A1S3EL69
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCH0ZCS4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73727
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410862584
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22318
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5PJB2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100128998
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6104
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01308
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID19123
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07453
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00749
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54676228
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DMC1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DMC0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCI3M072
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68293
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49157
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68292
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DMA8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID31378
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DMA6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DM92
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419492855

Total number of triples: 458.