http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AU-2006328424-B2

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filingDate 2006-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2013-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_570e9f8e49305b94bfc5c325a6f355e5
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publicationDate 2013-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AU-2006328424-B2
titleOfInvention Method of producing drug-containing wax matrix particles, extruder to be used in the method and sustained-release preparation containing cilostazol
abstract It is intended to provide a method of conveniently producing drug-containing wax matrix particles (in particular, drug-containing wax matrix particles having an average particle diameter of 1 mm or less) through melting and spraying steps without suffering from a jamming failure caused by the recrystallization of the once molten drug. Namely, drug-containing wax matrix particles containing a drug and a wax are produced via the following steps (i) and (ii): (i) the step of feeding the drug and wax as described above into an extruder wherein the temperatures of a barrel (1) and a die have been controlled to a level higher than the melting point of the wax; and (ii) the step of melt-kneading the drug with the wax in the extruder as described above and simultaneously spraying out the melt-kneaded mixture comprising the drug and the wax from a spray nozzle (5), which is attached directly to a die (3) provided at the tip of the barrel (1) in the extruder, into an atmosphere at a temperature lower than the melting point of the wax to thereby form particles.
priorityDate 2005-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 894.