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publicationDate 2018-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber AR-108245-A1
titleOfInvention SYNTHESIS OF INDAZOLES
abstract Claim 1: A method for preparing a compound of formula (1), characterized in that it comprises the following step (A): wherein a compound of formula (2) is allowed to react with a vinyl sulfone compound of formula (3), in the which R represents an alkyl group, such as a methyl, ethyl or n-propyl group for example, or an aryl group, such as a phenyl group for example, optionally in an aromatic hydrocarbon solvent, such as toluene for example, preferably at the reflux temperature of said solvent, thereby providing said compound of formula (1).
priorityDate 2016-04-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 50.