http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-106084-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_173bc2c63b34988699010ba05e5b1376 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D261-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D261-02 |
| filingDate | 2016-09-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9174c1b59f425844befe94addcd4446a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ce3fdd1c8c7ff1498cec412400ccf09a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b68c0009b74ac8c46a990903ecdce0aa http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_94659be065d70be2d9dc03a943b9c73a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0400a4cadc7d0fc991311ac00ded89a5 |
| publicationDate | 2017-12-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-106084-A1 |
| titleOfInvention | BENZAMIDS REPLACED WITH ISOXAZOLINE AS INSECTICIDES |
| abstract | Compounds and intermediates and stereoisomers, enantiomers, tautomers, N-oxides and agrochemically acceptable salts of these compounds, as well as their uses as insecticides. Claim 1: A compound of formula (1), wherein A¹, A², A³ and A⁴ are independently from each other, C-H, C-R⁵ or N; R¹ is hydrogen, formyl, C₁₋₈ alkyl, (C₁₋₈ alkyl) carbonyl-, C alco alkoxy, (C₁₋₈ alkoxy) - (C₁₋₈ alkoxy) carbonyl, phenyl- ( C₁₋₈ alkoxy) carbonyl, phenyl- (C₁₋₄ alkyl), phenyl- (C₁₋₄ alkyl) where the phenyl moiety is substituted with one to three R⁷; R² is hydrogen, halogen, cyano, C₁₋₈ alkyl or C₁₋₈ alkyl substituted with one to three R⁶ᵃ, haloalkyl C₁₋₈ or haloalkyl C₁₋₈ substituted with one to three R⁶ᵃ, cycloalkyl C₃₋₈ or cycloalkyl C₃₋ ₈ substituted with one to three R⁶ᵇ C₃₋₈ cycloalkyl where a carbon atom is replaced by O, S, S (O) or SO₂, or (C₃₋₈ cycloalkyl) - (C₁₋₈ alkyl), (C₃₋ cycloalkyl) ₈) - (C₁₋₈ alkyl) where a carbon atom in the cycloalkyl group is replaced by O, S, S (O) or SO₂, or (C₃₋₈ cycloalkyl) - (C₁₋₈ haloalkyl), C₂₋ alkenyl ₈ or C₂₋₈ alkenyl substituted with one to three R⁶ᵃ, C halo haloalkenyl or C₂₋₈ haloalkenyl substituted with one to three R⁶ᵃ, C₂₋₈ alkynyl, C₂₋₈ haloalkynyl, phenyl, phenyl substituted with one to three R⁷, phenyl- (C₁₋₄ alkyl), phenyl- (C₁₋₄ alkyl) where the phenyl moiety is substituted with one to three R⁷, 5-6 membered heteroaryl, 5-6 membered heteroaryl substituted with one to three R⁷, 5-6 membered heteroaryl- (C alquilo alkyl) or 5-6 membered heteroaryl- (C₁₋₄ alkyl) where the heteroaryl moiety is substituted with one to three R⁷, -NH (R⁸), -N (R⁸) (R⁹), -OR¹⁰, -SR¹⁰, -S (O) R¹⁰, -S (O) ₂R¹⁰, COR¹⁰, COOR¹⁰; R³ is C₁₋₈ haloalkyl; R⁴ is phenyl or phenyl substituted with one to three R⁶ᵇ, or pyridine or pyridine substituted with one to three R⁶ᵇ; R⁵ is independently halogen, cyano, nitro, C₁₋₈ alkyl, C₃₋₈ cycloalkyl, C₁₋₈ haloalkyl, C₂₋₈ alkenyl, C₂₋₈ haloalkenyl, C₂₋₈ alkynyl, C₂₋₈ haloalkynyl, C₁₋₈ alkoxy, haloalkoxy C₁₋₈ or (C₁₋₈ alkoxy) carbonyl-, or two R⁵ in adjacent carbon atoms together form a bridge -CH = CH-CH = CH- or a bridge -N = CH-CH = CH-; each R⁶ᵃ is independently halogen, cyano, nitro, amino, hydroxy, oxo, C₁₋₈ alkylamino, hydroxyimino, C₁₋₈ alkyloxyimino, di (C₁₋₈ alkyl) amino, C₁₋₈ alkoxy, acetyloxy, formyloxy, C₁₋₈ haloalkoxy , C₁₋₄ alkylthio or tri (C₁₋₄ alkyl) silyl; each R⁶ᵇ is independently halogen, cyano, nitro, C₁₋₈ alkyl, C₁₋₈ haloalkyl, amino, C₁₋₈ alkylamino, di (C₁₋₈ alkyl) amino, hydroxyl, C₁₋₄ alkylthio, C₁₋₈ alkoxy or C₁ haloalkoxy ₋₈; R⁷ is independently halogen, cyano, nitro, C₁₋₈ alkyl, C₁₋₈ haloalkyl, C₁₋₈ alkoxy or C₁₋₈ haloalkoxy; R⁸ and R⁹ are independently hydrogen, cyano, cyano- (C₁₋₈ alkyl), C₁₋₈ alkyl or C₁₋₈ alkyl substituted with one to three R⁶ᵃ, C₁₋₈ alkoxy, C₁₋₈ haloalkoxy, C₁₋₈ substituted haloalkoxy with one to three R⁶ᵃ, C alco alkoxy substituted with one to three R⁶ᵃ, C halo haloalkyl or C₁₋₈ haloalkyl substituted with one to three R⁶ᵃ, C₃₋₈ cycloalkyl or C₃₋₈ cycloalkyl substituted with one to three R⁶ᵇ, C₃₋₈ cycloalkyl where a carbon atom is replaced by O, S, S (O) or SO₂, or (C₃₋₈ cycloalkyl) - (C₁₋₈ alkyl), (C₃₋₈ cycloalkyl) - (alkyl C₁₋₈) where a carbon atom in the cycloalkyl group is replaced by O, S, S (O) or SO₂, or (C₃₋₈ cycloalkyl) - (C₁₋₈ haloalkyl), C₂₋₈ alkenyl or C₂₋ alkenyl ₈ substituted with one to three R⁶ᵃ, haloalkenyl C₂₋₈ or haloalkenyl C₂₋₈ substituted with one to three R⁶ᵃ, alkynyl C₂₋₈, C₂₋₈ haloalkynyl, phenyl, phenyl substituted with one to three R⁷, phenyl- (C₁₋₄ alkyl), phenyl- (C₁₋₄ alkyl) where the phenyl moiety is substituted with one to three R⁷, 5-6 membered heteroaryl, 5-6 membered heteroaryl substituted with one to three R⁷, (5-6 membered heteroaryl) - (C₁₋₄ alkyl) or (5-6 membered heteroaryl) - (C₁₋ alkyl ₄) where the heteroaryl moiety is substituted with one to three R⁷, or R⁸ and R⁹, together with the nitrogen atom, can be linked by a C₃₋₈ alkylene chain, a C₃₋₈ alkylene chain substituted with one to three R⁶ᵇ or a C₃₋₈ alkylene chain where a carbon atom is replaced by O, S, S (O) or SO₂; R¹⁰ is hydrogen, cyano, cyano- (C₁₋₈ alkyl), C₁₋₈ alkyl or C₁₋₈ alkyl substituted with one to three R⁶ᵃ, haloalkyl C₁₋₈ or haloalkyl C₁₋₈ substituted with one to three R⁶ᵃ, cycloalkyl C₃₋₈ or C₃₋₈ cycloalkyl substituted with one to three R⁶ᵇ, C₃₋₈ cycloalkyl where a carbon atom is replaced by O, S, S (O) or SO₂, or (C₃₋₈ cycloalkyl) - (C₁ alkyl ₋₈), (C₃₋₈ cycloalkyl) - (C₁₋₈ alkyl) where a carbon atom in the cycloalkyl group is replaced by O, S, S (O) or SO₂, or (C₃₋₈ cycloalkyl) - (haloalkyl C₁₋₈), C₂₋₈ alkenyl or C₂₋₈ alkenyl substituted with one to three R⁶ᵃ, C₂₋₈ haloalkenyl or C₂₋₈ haloalkenyl substituted with one to three R⁶ᵃ, C₂₋₈ alkynyl, C₂₋₈ haloalkynyl, phenyl , phenyl substituted with one to three R⁷, phenyl- (C₁₋₄ alkyl), phenyl- (C₁₋₄ alkyl) where the phenyl moiety is substituted co n from one to three R⁷, 5-6 membered heteroaryl, 5-6 membered heteroaryl substituted with one to three R⁷, (5-6 membered heteroaryl) - (C₁₋₄ alkyl) or (5-6 heteroaryl members) - (C₁₋₄ alkyl) where the heteroaryl moiety is substituted with one to three R⁷; and one of its salts, stereoisomers, enantiomers, tautomers and agrochemically acceptable N-oxides. Claim 8: A compound of formula (2) wherein A¹, A², A³, A⁴, R¹ and R² are as defined for a compound of formula (1) in any of claims 1-7 and XB is a halogen, such as bromine, or XB is cyano, formyl, CH = N-OH or acetyl; or one of its salts or N-oxides. Claim 9: A compound of formula (3) wherein A¹, A², A³, A⁴, R¹ and R² are as defined for a compound of formula (1) in any of claims 1-7 and XC is CH₂-halogen, CH = C (R³) R⁴ or CH₂C (OH) (R³) R⁴ where R³ and R⁴ are as defined for a compound of formula (1); or one of its salts or N-oxides. Claim 10: A compound of formula (4) wherein R¹ and R² are as defined for a compound of formula (1) in any of claims 1-7; or one of its salts or N-oxides. Claim 11: A compound of formula (5) wherein A¹, A², A³, A⁴, R¹, R³ and R⁴ are as defined for a compound of formula (1) in any of claims 1-7; or one of its salts or N-oxides. |
| priorityDate | 2015-09-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 40.