http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-106070-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_173bc2c63b34988699010ba05e5b1376 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D261-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D261-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-12 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D261-02 |
| filingDate | 2016-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ce3fdd1c8c7ff1498cec412400ccf09a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_94659be065d70be2d9dc03a943b9c73a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9174c1b59f425844befe94addcd4446a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0400a4cadc7d0fc991311ac00ded89a5 |
| publicationDate | 2017-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-106070-A1 |
| titleOfInvention | BENZAMIDS REPLACED WITH ISOXAZOLINE AS INSECTICIDES |
| abstract | The present application refers to compounds, intermediates, compositions and methods of use. Claim 1: A compound of formula (1) wherein A¹, A², A³ and A⁴ are independently from each other C-H, C-R⁵, or nitrogen; R¹ is hydrogen, C₁₋₈ alkyl, C₁₋₈- alkylcarbonyl, C₁₋₈ alkoxy, C₁₋₈ alkoxy-C₁₋₈ alkyl or C₁₋₈- alkoxycarbonyl; R² is C₁₋₈ alkyl, C₁₋₈ alkyl substituted with one to three R⁶ᵃ, C₁₋₈ haloalkyl, C₁₋₈ haloalkyl substituted with one to three R⁶ᵃ, C₃₋₈ cycloalkyl, C₃₋₈ cycloalkyl substituted with one to three R⁶ᵇ, C₃₋₈ cycloalkyl where a carbon atom is replaced by O, S, S (O) or SO₂, C₃₋₈ cycloalkyl-C₁₋₈ alkyl, C₃₋₈ cycloalkyl-C₁₋₈ alkyl where a carbon atom in the group Cycloalkyl is replaced by O, S, S (O) or SO₂, C₃₋₈-C halo-haloalkyl, C₂₋₈ alkenyl, C₂₋₈ alkenyl substituted with one to three R⁶ᵃ, C₂₋₈ haloalkenyl, C₂₋₈ haloalkenyl substituted with one to three R⁶ᵃ, Cin alkynyl, C₂₋₈ haloalkynyl, phenyl, phenyl substituted with one to three R⁷, phenyl-C₁₋₄ alkyl, phenyl-C₁₋₄ alkyl wherein the phenyl moiety is substituted with one to three R⁷, 5-6 membered heteroaryl, substituted 5-6 membered heteroaryl with one to three R⁷, heteroaryl-C₁₋₄ alkyl of 5-6 members, heteroaryl-C₁₋₄ alkyl of 5-6 members wherein the heteroaryl moiety is substituted with one to three R-, -N (R⁸) (R⁹) , halogen or -OR¹⁰; R³ is C₁₋₈ haloalkyl; R⁴ is aryl, aryl substituted with one to three R⁷, heteroaryl or heteroaryl substituted with one to three R⁷; R⁵ is independently halogen, cyano, nitro, C₁₋₈ alkyl, C₃₋₈ cycloalkyl, C₁₋₈ haloalkyl, C₂₋₈ alkenyl, C₂₋₈ haloalkenyl, C₂₋₈ alkynyl, C₂₋₈ haloalkynyl, C₁₋₈ alkoxy, haloalkoxy C₁₋₈ or C₁₋₈- alkoxycarbonyl, or two R⁵ in adjacent carbon atoms together form a bridge -CH = CH-CH = CH- or a bridge -N = CH-CH = CH-; R⁶ᵃ is independently cyano, nitro, amino, C₁₋₈ alkylamino, N, N-C-dialkylamino, hydroxy, C₁₋₈ alkoxy or C₁₋₈ haloalkoxy; R⁶ᵇ is independently halogen, cyano, nitro, oxo, C₁₋₈ alkyl, C₁₋₈ haloalkyl, amino, C₁₋₈ alkylamino, N, N-C-dialkylamino, hydroxyl, C₁₋₈ alkoxy, C₁₋₈ haloalkoxy, phenyl , phenyl substituted with one to three R⁷, 5-6 membered heteroaryl, 5-6 membered heteroaryl substituted with one to three R⁷; R⁷ is independently halogen, cyano, nitro, C₁₋₈ alkyl, C₁₋₈ haloalkyl, C₁₋₈ alkoxy, C₁₋₈ haloalkoxy; R⁸ and R⁹ are independently hydrogen, cyano, cyano-C₁₋₈ alkyl, C₁₋₈ alkyl, C₁₋₈ alkyl substituted with one to three R⁶ᵃ, C₂₋₈ alkenyl, C₂₋₈ alkenyl substituted with one to three R⁶ᵃ, C₁ alkoxy ₋₈, C₁₋₈ haloalkoxy, C₁₋₈ haloalkoxy substituted with one to three R⁶ᵃ, C₁₋₈ alkoxy substituted with one to three R⁶ᵃ, haloalkyl C₁₋₈, haloalkyl C₁₋₈ substituted with one to three R⁶ᵃ, cycloalkyl C₃₋₈ , C₃₋₈ cycloalkyl substituted with one to three R⁶ᵇ, C₃₋₈ cycloalkyl where a carbon atom is replaced by O, S, S (O) or SO₂, C₃₋₈ cycloalkyl-C₁₋₈ alkyl, C₃₋₈- cycloalkyl C₁₋₈ alkyl where a carbon atom in the cycloalkyl group is replaced by O, S, S (O) or SO₂, C₃₋₈ cycloalkyl-C₁₋₈ haloalkyl, C₂₋₈ alkenyl, C₂₋₈ alkenyl substituted with one to three R⁶ᵃ, haloalkenyl C₂₋₈, haloalkenyl C₂₋₈ substituted c on one to three R⁶ᵃ, C₂₋₈ alkynyl, C₂₋₈ haloalkynyl, phenyl, phenyl substituted with one to three R⁷, phenyl-C₁₋₄ alkyl, phenyl-C₁₋₄ alkyl wherein the phenyl moiety is substituted with one to three R⁷, 5-6 membered heteroaryl, 5-6 membered heteroaryl substituted with one to three R⁷, 5-6 membered heteroaryl-C, alkyl, 5-6 membered heteroaryl-alkyl wherein the heteroaryl moiety is substituted with one to three R⁷, -S (O) R¹⁰, -S (O) ₂R¹⁰, COR¹⁰, COOR¹⁰, or R⁸ and R⁹ together with the nitrogen atom can be linked through a C₃₋₈ alkylene chain, a chain C₃₋₈ alkylene substituted with one to three R⁶ᵇ or a C₃₋₈ alkylene chain, where a carbon atom is replaced by O, S, S (O) OR SO₂; R¹⁰ is hydrogen, cyano-C₁₋₈ alkyl, C₁₋₈ alkyl, C₁₋₈ alkyl substituted with one to three R⁶ᵃ, haloalkyl C₁₋₈, haloalkyl C₁₋₈ substituted with one to three R⁶ᵃ, cycloalkyl C₃₋₈, cycloalkyl C₃ ₋₈ substituted with one to three R⁶ᵇ, C₃₋₈ cycloalkyl where a carbon atom is replaced by O, S, S (O) or SO₂, C₃₋₈ cycloalkyl-C₁₋₈ alkyl, C₃₋₈ cycloalkyl-C alquilo alkyl ₈ where a carbon atom in the cycloalkyl group is replaced by O, S, S (O) or SO₂, C₃₋₈-Cal-haloalkyl, Cal alkenyl, Cque alkenyl substituted with one to three R⁶ᵃ, C₂₋₈ haloalkenyl, C₂₋₈ haloalkenyl substituted with one to three R⁶ᵃ, C₂₋₈ alkynyl, C₂₋₈ haloalkynyl, phenyl, phenyl substituted with one to three R⁷, phenyl-C₁₋₄ alkyl, phenyl-C₁₋₄ alkyl in where the phenyl moiety is substituted with one to three R⁷, 5-6 membered heteroaryl, 5-6 membered heteroaryl substituted with one to three R⁷, 5-6 membered heteroaryl-C o alkyl or 5-6 membered heteroaryl-alkyl wherein the heteroaryl moiety is substituted with one to three R⁷; n is 1 or 2; or a tautomer, isomer, enantiomer, salt or N-oxide thereof. Claim 10: A compound of formula (2) wherein A¹, A², A³, A⁴, R¹ and R² are as defined for a compound of formula (1) according to any one of claims 1 to 9 and XB it is a leaving group, or XB is cyano, formyl, CH = N-OH or acetyl; or a tautomer, isomer, enantiomer, salt or N-oxide thereof; or a compound of formula (3) wherein A¹, A², A³, A⁴, R¹ and R², are as defined for a compound of formula (1) according to any one of claims 1 to 9 and XC is CH₂ -halogen, CH = C (R³) R⁴ or CH₂C (OH) (R³) R⁴ wherein R³ and R⁴ are as defined for a compound of formula (1) according to any one of claims 1 to 9; or a tautomer, isomer, enantiomer, salt or N-oxide thereof; or a compound of formula (4) wherein R¹ and R² are as defined for a compound of formula (1) according to any one of claims 1 to 9; or a tautomer, isomer, enantiomer, salt or N-oxide thereof. |
| priorityDate | 2015-09-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 33.