http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-098626-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_981a37900e6991fb373304ed2ba5a703 |
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C2601-02 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C47-546 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C47-55 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C25-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C47-575 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N35-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C47-542 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-44 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C211-17 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N33-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N29-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C22-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-12 |
| filingDate | 2014-12-05-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bb9dc67551d50d5bab43b4745f30f64c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_04d477d12520ae748237962623bdd30b http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8f9838d8c2ecd0318dd1c3d6626b40b2 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8e7b92ad7043071b45a7b55b54f5d7f7 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8dee7c05b59a65298d03651065a0704a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a1354c42cab65e86c9b68204870ecb70 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_320af7db0f549f3f9ae53065a3e26ead http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8ce43c126ccd053e4df78924e4255054 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_dda4f1af430ef42b0f2d4ecda577c0b1 |
| publicationDate | 2016-06-01-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-098626-A1 |
| titleOfInvention | DERIVATIVES OF N-CICLOALQUIL-N - {[2- (1-CICLOALQUIL REPLACED) PHENYL] METHYLENE} - (UNCLE) CARBOXAMIDE |
| abstract | This refers to fungicidal derivatives of N-cycloalkyl-N - {[2- (substituted 1-cycloalkyl) phenyl] methylene} carboxamide and their thiocarbonyl derivatives, their preparation processes and intermediate compounds for their preparation, use as fungicides, particularly in the form of fungicidal compositions and methods for the control of plant pathogenic fungi using these compounds or their compositions. Claim 1: A compound of formula (1) wherein X¹ and X² which may be the same or different, represent a chlorine or fluorine atom; T represents O or S; n represents 0, 1, 2, 3 or 4; m represents 0, 1, 2, 3, 4, 5 or 6; p represents 1, 2, 3, 4 or 5; Z¹ represents an unsubstituted C₃₋₇ cycloalkyl or a C₃₋₇ substituted cycloalkyl with up to 10 atoms or groups that may be the same or different and that may be selected from the list consisting of halogen, cyano, C₁₋₈ alkyl, halogenoalkyl atoms C₁₋₈ comprising up to 9 halogen atoms that may be the same or different, C₁₋₈ alkoxy, C₁₋₈ halogenalkoxy comprising up to 9 halogen atoms that may be the same or different, C₁₋₈ carbonyl alkoxy, C₁₋₈ halogenalkoxy carbonyl comprising up to 9 halogen atoms that may be the same or different, C₁₋₈-aminocarbonyl alkyl and di-C₁₋₈-aminocarbonyl alkyl; Z² and Z³, which may be the same or different, represent a hydrogen atom; C₁₋₈ substituted or unsubstituted alkyl; C₂₋₈ substituted or unsubstituted alkenyl; C₂₋₈ substituted or unsubstituted alkynyl; cyano; isonitrile; nitro; a halogen atom; C₁₋₈ substituted or unsubstituted alkoxy; C₂₋₈ substituted or unsubstituted alkenyloxy; C₂₋₈ substituted or unsubstituted alkynyloxy; C₃₋₇ substituted or unsubstituted cycloalkyl; C₁₋₈-substituted or unsubstituted alkyl sulfanyl; C₁₋₈-substituted or unsubstituted alkyl sulfonyl; C₁₋₈-substituted or unsubstituted alkyl sulfinyl; Not me; C₁₋₈-substituted or unsubstituted alkyl amino; Cquil-substituted or unsubstituted dialkyl amino; C₁₋₈ substituted or unsubstituted C alkoxy; C₁₋₈-alkyl substituted or unsubstituted carbamoyl; dialkyl C₁₋₈ substituted or unsubstituted carbamoyl; or substituted or unsubstituted C₁₋₈-C₁₋₈-alkoxy C-alkoxy; or Z² and Z³ together with the carbon atom to which they are attached can form a substituted or unsubstituted C₃₋₇ cycloalkyl; Z⁴ represents a halogen atom; hydroxy; cyano; C₁₋₈ substituted or unsubstituted alkyl; C₁₋₈ halogenalkyl having 1 to 5 halogen atoms; C₂₋₈ substituted or unsubstituted alkenyl; C₂₋₈ halogenoalkenyl having 1 to 5 halogen atoms; C₂₋₈ substituted or unsubstituted alkynyl; C₂₋₈ halogenoalkynyl having 1 to 5 halogen atoms; C₁₋₈ substituted or unsubstituted alkoxy; C₁₋₈ halogenoalkoxy having 1 to 5 halogen atoms; C₁₋₈-substituted or unsubstituted alkyl sulfanyl; formyl; C₁₋₈ alkyl substituted or unsubstituted; carboxy; or C₁₋₈ substituted or unsubstituted C alkoxy; W independently represents a halogen atom; nitro; cyano; isonitrile; hydroxy; Not me; sulfanyl; pentafluoro-l⁶-sulfanyl; formyl; formyloxy; formylamino; (hydroxyimino) -C₁₋₈ substituted or unsubstituted alkyl; (C₁₋₈ alkoxyimino) -C₁₋₈ substituted or unsubstituted alkyl; (C₂₋₈imino alkenyloxy) -C₁₋₈ substituted or unsubstituted alkyl; (C₂₋₈imino alkynyloxy) -C₁₋₈ substituted or unsubstituted alkyl; (benzyloxyimino) -C₁₋₈ substituted or unsubstituted alkyl; carboxy; carbamoyl; N-hydroxycarbamoyl; carbamate; C₁₋₈ substituted or unsubstituted alkyl; C₁₋₈ halogenalkyl having 1 to 9 halogen atoms; C₂₋₈ substituted or unsubstituted alkenyl; C₂₋₈ halogenoalkenyl having 1 to 9 halogen atoms; C₂₋₈ substituted or unsubstituted alkynyl; C₂₋₈ halogenoalkynyl having 1 to 9 halogen atoms; C₁₋₈ substituted or unsubstituted alkoxy; C₁₋₈ halogenoalkoxy having 1 to 9 halogen atoms; C₁₋₈-substituted or unsubstituted alkyl sulfanyl; halogen C₁₋₈ sulfanyl alkyl having 1 to 9 halogen atoms; C₁₋₈-substituted or unsubstituted alkyl sulfinyl; halogen C₁₋₈ sulfinyl alkyl having 1 to 9 halogen atoms; C₁₋₈-substituted or unsubstituted alkyl sulfonyl; halogen C₁₋₈ sulfonyl alkyl having 1 to 9 halogen atoms; C₁₋₈-substituted or unsubstituted alkyl amino; Cquil-substituted or unsubstituted dialkyl amino; C₂₋₈ substituted or unsubstituted alkenyloxy; C₂₋₈ halogenoalkenyloxy having 1 to 9 halogen atoms; C₃₋₈ substituted or unsubstituted alkynyloxy; C₂₋₈ halogenoalkyloxy having 1 to 9 halogen atoms; C₃₋₇ substituted or unsubstituted cycloalkyl; C₃₋₇ halocycloalkyl having 1 to 9 halogen atoms; (C₃₋₇ cycloalkyl) -C₁₋₈ substituted or unsubstituted alkyl; C₄₋₇ substituted or unsubstituted cycloalkenyl; C₄₋₇ halogenocycloalkenyl having 1 to 9 halogen atoms; (C₃₋₇-cycloalkyl) -C no substituted or unsubstituted alkenyl; (C₃₋₇-cycloalkyl) -C₂₋₈ substituted or unsubstituted alkynyl; bicyclo [2.2.1] substituted or unsubstituted heptanyl; bicyclo [2.2.1] substituted or unsubstituted heptenyl; tri (C₁₋₈) alkyl substituted or unsubstituted silyl; tri (C₁₋₈ alkyl) silyl substituted or unsubstituted C₁₋₈ alkyl; C₁₋₈ alkyl substituted or unsubstituted; halogen C₁₋₈ carbonyl alkyl having 1 to 9 halogen atoms; C₁₋₈ alkyl substituted or unsubstituted carbonyloxy; halogen C₁₋₈ carbonyloxy alkyl having 1 to 9 halogen atoms; C₁₋₈ alkyl substituted or unsubstituted carbonylamino; halogen C₁₋₈ carbonylamino alkyl having 1 to 9 halogen atoms; C₁₋₈ substituted or unsubstituted C alkoxy; Cógeno carbonyl halogenoalkoxy having 1 to 9 halogen atoms; C₁₋₈ alkyloxy substituted or unsubstituted; C₁₋₈ carbonyloxy halogenoalkoxy having 1 to 9 halogen atoms; C₁₋₈-alkyl substituted or unsubstituted carbamoyl; dialkyl C₁₋₈ substituted or unsubstituted carbamoyl; substituted or unsubstituted C₁₋₈-aminocarbonyloxy alkyl; substituted or unsubstituted Cquil-aminocarbonyloxy; N- (C₁₋₈-alkyl) substituted or unsubstituted hydroxycarbamoyl; C₁₋₈ carbamoyl substituted or unsubstituted alkoxy; N- (C₁₋₈-alkyl) -C₁₋₈-substituted or unsubstituted C-carbamoyl; aryl that may be substituted by up to 6 Q groups that may be the same or different; C₁₋₈ arylalkyl which may be substituted by up to 6 Q groups that may be the same or different; C₂₋₈ arylalkenyl which may be substituted by up to 6 Q groups that may be the same or different; C₂₋₈ arylalkynyl which may be substituted by up to 6 Q groups that may be the same or different; aryloxy which may be substituted by up to 6 Q groups that may be the same or different; arylsulfanyl which may be substituted by up to 6 Q groups that may be the same or different; arylamino which may be substituted by up to 6 Q groups that may be the same or different; C₁₋₈ arylalkyloxy which may be substituted by up to 6 Q groups that may be the same or different; C₁₋₈ arylalkyl sulfanyl which may be substituted by up to 6 Q groups that may be the same or different; C₁₋₈ arylalkylamino which may be substituted by up to 6 Q groups that may be the same or different; C₁₋₈ heteroarylalkyl which may be substituted by up to 6 Q groups that may be the same or different; heteroaryl which may be substituted by up to 4 Q groups; or heteroaryloxy which may be substituted by up to 4 Q groups; or Z⁴ and its neighboring substituent W, together with the carbon atom to which they are attached, can form a substituted or unsubstituted C₄₋₇ cycloalkyl; Y independently represents a halogen atom; C₁₋₈ alkyl; C₁₋₈ halogenalkyl having 1 to 9 halogen atoms; C₁₋₈ substituted or unsubstituted alkoxy; C₁₋₈ halogenoalkoxy having 1 to 9 halogen atoms; C₁₋₈-substituted or unsubstituted alkyl sulfanyl; halogen C₁₋₈ sulfanyl alkyl having 1 to 9 halogen atoms; or C₁₋₈ substituted or unsubstituted C alkoxy; Q independently represents a halogen, cyano, nitro, substituted or unsubstituted C₁₋₈ alkyl, C₁₋₈ halogen alkyl comprising up to 9 halogen atoms that may be the same or different, C₁₋₈ substituted or unsubstituted alkoxy, C₁ halogenalkoxy ₋₈ comprising up to 9 halogen atoms that may be the same or different, substituted or unsubstituted C₁₋₈ alkyl sulfanyl, C₁₋₈ halogenoalkylsulfanyl comprising up to 9 halogen atoms that may be the same or different, tri (C₁₋₈ alkyl) substituted or unsubstituted silyl, tri (C₁₋₈ alkyl) silyl substituted or unsubstituted C₁₋₈ alkyl, (C₁₋₈imino alkoxy) -substituted or unsubstituted C₁₋₈alkyl, or (benzyloxyimino) -C₁₋₈ alkyl substituted or unsubstituted; in addition to its salts, N-oxides, metal complexes, metalloid complexes and optically active isomers or geometric isomers thereof. Claim 13: A compound of formula (2), in addition to its acceptable salts, wherein Z¹, Z², Z³, Z⁴, n, m, p, W and Y are as defined in any one of claims 1 to 12. Claim 14: A compound of formula (3) wherein Z⁴, n, m, p, W and Y are as defined in any of claims 1 to 12, provided that compound of formula (3) does not represent: 2- (1-Methoxycycloheptyl) -5- (trifluoromethyl) benzaldehyde, (1S, 2S) -2-ethoxy-2- (2-formylphenyl) cyclopropanecarboxylate, and (1S, 2R) -2-ethoxy-2- (2- methyl formylphenyl) cyclopropanecarboxylate. Claim 15: A compound of formula (4), wherein U² is a halogen and Z⁴, n, m, p, W and Y are as defined herein, provided that the compound of formula (4) does not represent: 1- [2- (bromomethyl) -3-chlorophenyl] cyclobutanol, 1- [2- (bromomethyl) phenyl] cyclopropanecarbonitrile, 1- [2- (bromomethyl) -4- (trifluoromethyl) phenyl] cycloheptyl methyl ether, 2- (bromomethyl) -1- (1-methoxycyclopentyl) -4- (trifluoromethyl) benzene, 2- (bromomethyl) -1- (1-methoxycyclohexyl) -4- (trifluoromethyl) benzene, and 1- [2- (bromomethyl) phenyl] cyclopentanecarbonitrile. |
| priorityDate | 2013-12-05-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 78.