http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-094112-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_5257f76a7c47cfed7f46b0cb9994e6a8 |
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| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-40 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D307-36 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C235-70 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N37-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D331-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C237-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C233-57 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C233-01 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D213-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D309-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D305-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D261-12 |
| filingDate | 2013-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_56a73d7134f5c1707aa3d72a9443611d http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_81930d3e696fb695370bdd596bcf2585 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c049d61f138ebc652acfdee3658a81a4 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_d1ec82f41c2b49691286448b86dbd44c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_efa368294bceae989df84da19edfb220 |
| publicationDate | 2015-07-08-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-094112-A1 |
| titleOfInvention | (HETERO) USEFUL ARILACRILAMIDS TO CONTROL ECTOPARASITOS |
| abstract | Claim 1: A compound characterized in that it is of formula (1), including all geometric isomers and stereoisomers, N-oxides, S-oxides, salts and prodrugs thereof, wherein T¹, T² and T³ are independently of each other C ( R⁰) or is N, where the amount of nitrogen atoms in T¹-T³ is between 0 and 2; R⁰ is H or R¹; n is 1, 2 or 3; R¹ is halogen, cyano (-CN), nitro (-NO₂), C₁₋₆ alkyl, C₃₋₆ cycloalkyl, C₂₋₆ alkenyl, C₂₋₆ alkynyl, C₁₋₆ haloalkyl, C₁₋₆ alkoxy, C₁₋₆ haloalkoxy , C₁₋₆thio alkyl, C₁₋₆thio haloalkyl, C₁₋₆sulfinyl alkyl, C₁₋₆sulfinyl haloalkyl, C₁₋₆sulfonyl alkyl, C₁₋₆sulfonyl haloalkyl, N-mono- or N, N-di-C₁₋₆amino alkyl, C₁₋ alkoxy Boncarbonyl, C₁₋₆carbonyl alkyl, aminosulfonyl, C₁₋₆aminosulfonyl alkyl, C₁₋₆sulfonylamino alkyl or phenyl which is unsubstituted or substituted by halogen, cyano, nitro, C₁₋₄ haloalkyl, C₁₋₄ haloalkoxy or C₁₋₄thio haloalkyl; or R¹ is a carbon chain C₁₋₄ that optionally contains 1-2 heteroatoms of the group of N, S, O, which joins two adjacent ring positions and forms an aliphatic, aromatic, heteroaromatic or heterocyclic ring that is optionally monosubstituted or polysubstituted with C₁₋₆ alkyl or halogen, in which case n is 2; X is C₁₋₆ alkyl, C₁₋₄ alkoxy-C₁₋₆ alkyl, C₁₋₆carbonyl alkoxy, C₁₋₆ haloalkyl, C₃₋₆ cycloalkyl or C₃₋₆ halocycloalkyl; R² is hydrogen, cyano, hydroxyl, C₁₋₆ alkyl, C₂₋₆ alkenyl, C₂₋₆ alkynyl, C₁₋₆ alkoxy or C₃₋₆ cycloalkyl; R³ is hydrogen, C₁₋₆ alkyl or C₁₋₆carbonyl alkyl; R⁴ and R⁵ are independently hydrogen, halogen, C₁₋₆ alkyl or C₁₋₆ alkoxy; And it is a radical selected from the group of formulas (2), where the second connection site (right) in each case is connected to unit C (O) NR⁷R⁸; m is the integer 0, 1 or 2; m1 is the integer 0 or 1; R⁶ is halogen, cyano, nitro, C₁₋₆ alkyl, C₂₋₆ alkenyl, C₂₋₆ alkynyl, C₃₋₆ cycloalkyl, C₄₋₇ alkylcycloalkyl, C₄₋₇ cycloalkylalkyl, C₁₋₆ alkoxy, C₁₋₆carbonyl alkyl C₁₋₆carbonyl alkoxy; A is an anelated 5 or 6 membered heteroaromatic ring comprising T⁸; T⁴ is S or O; T⁵ is N, CH or C (CH₃); T⁶ and T⁷ are independently of each other CH or N where the amount of nitrogen atoms in T⁶-T⁷ is 0 or 1; T⁸ is N or O; R⁷ is H, C₁₋₆ alkyl which is unsubstituted or substituted by halogen, C₁₋₄ alkoxy, C₁₋₂thio alkyl, cyano, nitro, amino or N-mono- or N, N-di-C₁₋₄amino alkyl, or is C₂₋₄ alkenyl, C₂₋₄ alkynyl or C₃₋₆ cycloalkyl; R⁸ is H; a group -CH = N-OR⁹; a radical Q; a radical Q¹; or is C₁₋₆ alkyl, C₂₋₆ alkenyl, C₂₋₆ alkynyl, C₃₋₆ cycloalkyl, C₄₋₇ alkylcycloalkyl, C₄₋₇ cycloalkylalkyl, C₅₋₁₀ bicyclo-alkylene or C₃₋₆ cycloalcanone which in each case does not is substituted or substituted in the alkyl, cycloalkyl, alkenyl or alkynyl unit with halogen, hydroxy, carboxy (COOH), C₁₋₄ alkyl, C₁₋₆ alkoxy, haloC₁₋₆ alkoxy, C₁₋₆thio alkyl, C₁₋ haloalkyl ₆thio, C₁₋₆sulfinil alkyl, C₁₋₆sulfonyl alkyl, cyano, nitro, amino, N-mono- or N, N-di-C₁₋₆amino alkyl, C₃₋₆amino cycloalkyl, C₁₋₆carbonyl alkoxy, C₂₋₆carbonyl alkyl, alkyl C₁₋₆carbonylamino, aminosulfonyl, N-mono- or N, N-di-C₁₋₄aminosulfonyl alkyl, a group -C (W) NR⁹R¹⁰ or a radical Q; or R⁷ and R⁸ together are a group = C (R¹¹) -NR¹²R¹³ or = C (R¹¹) -C (NH₂) -OR¹²); or R⁷ and R⁸ together with the N atom to which they are attached, form a 3- and 7-membered ring that optionally contains an additional heteroatom selected from the group consisting of N, S and O, and where the ring is not substituted additionally or is mono-substituted or polysubstituted with C₁₋₂ alkyl, C₁₋₂ haloalkyl, C₁₋₂ alkoxy, hydroxy, halogen, cyano, nitro, N, N-di-C₁₋₂aminomethyl alkyl or N, N-di-C₁₋ alkyl ₂ aminocarbonylmethyl; Q and Q are independently of each other a C₆₋₁₀ aryl, a 4, 5, or 6 membered aliphatic or aromatic heterocyclic ring, or an 8, 9 or 10 membered aliphatic or aromatic fused heterobicyclic ring, where each of they are not substituted or are mono-substituted or polysubstituted with halogen, hydroxy, C₁₋₆ alkyl, C₂₋₆ alkenyl, C₂₋₆ alkynyl, C₃₋₆ cycloalkyl, C₃₋₆ cycloalkyl-C₁₋₂ alkyl, C₁₋₆ haloalkyl, C₁₋₆ alkoxy, C₁₋₆ haloalkoxy, C₁₋₆tio alkyl, C₁₋₆sulfinyl alkyl, C₁₋₆sulfonyl alkyl, cyano, nitro, amino, N-mono- or N, N-di-C₁₋₆amino alkyl, C₃₋ cycloalkyl ₆amino, COOH, C₁₋₆-carbonyl alkoxy, C₂₋₆carbonyl alkyl, C₁₋₆carbonylamino alkyl, aminocarbonyl, N-mono- or N, N-di-C₁₋₆aminocarbonyl alkyl, aminosulfonyl, N-mono- or N, N- di-C₁₋₄-amino sulfonyl alkyl, phenyl-C₁₋₄-alkyl unsubstituted or substituted by halogen or nitro, 5- or 6-membered heterocyclyl-C alquilo alkyl or a Q radical; Q is a C₆₋₁₀ carbocyclic ring or a 4, 5 or 6-membered heterocyclic ring, where each one is aromatic or not, where each of them is unsubstituted or is mono-substituted or polysubstituted with halogen, hydroxy, C₁₋₆ alkyl, C₂₋₆ alkenyl, C₂₋₆ alkynyl, C₃₋₆ cycloalkyl, C₁₋₆ haloalkyl, C₁₋₆ alkoxy, C₁₋₆thio alkyl, C₁₋₆sulfinyl alkyl, C₁₋₆sulfonyl alkyl, cyano, nitro, amino, N-mono- or N, N-di-C₁₋₆amino alkyl, C₃₋₆amino cycloalkyl, COOH, C₁₋₆carbonyl alkoxy, C₂₋₆carbonyl alkyl, C₁₋₆carbonylamino alkyl, aminocarbonyl, N-mono- or N, N-di-C₁₋₆-aminocarbonyl, aminosulfonyl, or N-mono- or N, N-di-C₁₋₄-amino-sulfonyl alkyl; Q¹ is a radical of formula (3), where Z is O or CH₂ and R¹⁴ is H, C₁₋₄ alkyl, or C₁₋₄ haloalkyl; R⁹ is H or C₁₋₆ alkyl; R¹⁰ is H, C₁₋₆ alkyl, C₂₋₆ alkenyl, C₂₋₆ alkynyl, C₃₋₆ cycloalkyl, C₄₋₇ alkylcycloalkyl or C₄₋₇ cycloalkylalkyl, which in each case is not substituted or substituted in the alkyl unit , alkenyl, alkynyl or cycloalkyl with halogen, cyano, nitro, hydroxy, carboxy (COOH), C₁₋₆ alkoxy, C halo haloalkoxy, C₁₋₆thio alkyl, C₁₋₆thio haloalkyl, C₁₋₆sulfinyl alkyl, C₁₋₆sulfonyl alkyl, amino, N-mono- or N, N-di-C₁₋₆amino alkyl, C₃₋₆amino cycloalkyl, C₁₋₆carbonyl alkoxy, C₂₋₆carbonyl alkyl, C₁₋₆carbonylamino alkyl, aminocarbonyl, N-mono- or N, N-di -C-amino-carbonyl, aminosulfonyl, N-mono- or N, N-di-C-amino-sulfonyl alkyl or a Q radical; R¹¹ is H C₁₋₆ alkyl or C₁₋₆ alkoxy; R¹² and R¹³ are independently of each other C alquilo alkyl; and W and W are independently of each other O or S. |
| priorityDate | 2012-12-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 86.