http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-081642-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_f2d3599fb8f8f479dba95ca9bb504884 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-5517 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P31-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-5517 |
| filingDate | 2011-06-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2012-10-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-081642-A1 |
| titleOfInvention | DERIVATIVES 5,6-DIHIDRO-4 - [(DIFLUOR-ETIL) PHENYL] -4H-PIRROLO [1,2-A] [1,4] BENZODIACEPIN AND 4- (DIFLUORETIL) PHENYL-6H-PIRROLO [1,2- A] [1,4] ANTIFUNGAL BENZODIACEPIN AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| abstract | The compounds according to the present are mainly active against dermatophytes and systemic fungal infections. This also relates to processes for the preparation of said compounds, pharmaceutical compositions comprising said compounds as an active ingredient as well as the use of said compounds as medicaments. Claim 1: A compound of formula (1) or a stereoisomeric form thereof. , where R1 is hydrogen, chlorine or fluorine; R2 is hydrogen, chlorine, fluorine or methyl; R3 and R4 are hydrogen; or R3 and R4 taken together form a bond; R5 is 1,1-difluoroethyl, and R6 is hydrogen or fluorine; or R5 is hydrogen or fluorine, and R6 is 1,1-difluoroethyl; or a pharmaceutically acceptable addition or solvate salt thereof. |
| priorityDate | 2010-06-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 23.