http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-077382-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_8e0bf0928b608797b70bbc2b91c7e52e |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N53-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-14 |
| filingDate | 2010-07-05-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2011-08-24-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-077382-A1 |
| titleOfInvention | PIRIDAZINE COMPOUNDS TO CONTROL INVERTEBRATE PESTS |
| abstract | A method for controlling invertebrate pests, a method for protecting plant propagation material and / or plants that grow from it, plant propagation material, which comprises at least one compound according to the present invention, a method for treating or protect an animal from infestation or infection by parasites and an agricultural composition that contains at least one compound according to the present invention. Claim 1: Pyridazine compounds characterized in that they have formulas 1 or 2: wherein A is an isoxazole or isothiazole radical of formulas A1, A2 or A3, wherein it indicates the binding site with the rest of formulas 1 or 2 , and where Z is O or S; R41, R42, R43 and R51 are independently selected from hydrogen, halogen, CN, NO2, C1-10 alkyl, C2-10 alkenyl and C2-10 alkynyl, wherein the last 3 radicals mentioned may be unsubstituted, they can be partially or totally halogenated or they can have 1, 2 or 3 identical or different Rx substituents, or where R41, R42, R43 and R51 are also selected from ORa, C (Y) Rb, C (Y) ORC, S ( O) mRd, NReRf, heterocyclyl, heteroaryl, C3-10 cycloalkyl, C5-10 cycloalkenyl and phenyl, wherein the last 5 radicals mentioned may be unsubstituted or may have 1, 2, 3, 4 or 5 identical or different Rx substituents ; R52, R53 are selected from hydrogen, halogen, CN, NO2, C1-10 alkyl, C2-10 alkenyl and C2-10 alkynyl, wherein the last 3 radicals mentioned may be unsubstituted, may be partially or totally halogenated or may have 1, 2 or 3 identical or different Rx substituents, or wherein R52, R53 are also selected from ORa, C (Y) Rb, C (Y) ORc, S (O) mRd, NReRf, heterocyclyl, heteroaryl, C3- cycloalkyl 10, C5-10 cycloalkenyl and phenyl, wherein the last 5 radicals mentioned may be unsubstituted or may have 1, 2, 3, 4 or 5 identical or different Rx substituents, and wherein V is C (Rv) or N; W is C (RW) or N; provided that V or W is N; Rt, Ru, Rv and Rw are independently selected from hydrogen, halogen, C1-4 alkyl, C1-3 haloalkyl, C1-4 alkoxy, C1-3 haloalkoxy, C1-4 alkylthio, C1-3 haloalkylthio, alkylsulfinyl C1-4, C1-3 haloalkylsulfinyl, C1-4 alkylsulfonyl, C1-3 haloalkylsulfonyl, C3-6 cycloalkyl, C3-6 halocycloalkyl, C2-4 alkenyl, C2-4 haloalkenyl, C2-4 alkynyl or C1-4 alkoxy C1-4; X1 is S, O or NR1a wherein R1 is selected from hydrogen, C1-10 alkyl, C1-4 haloalkyl, C3-10 cycloalkyl, C3-10 cycloalkylmethyl, C3-10 halocycloalkyl, C2-10 alkenyl, C2-10 haloalkenyl, C2-10 alkynyl, C1-10 alkoxy-C1-4 alkyl, phenyl, heteroaryl, heterocyclyl, phenyl-C1-4 alkyl, heteroaryl-C1-4 alkyl, heterocyclyl-C1-4 alkyl, wherein the ring, in the latter 6 mentioned radicals, can be unsubstituted or can have 1, 2, 3, 4 or 5 substituents that are selected, independently from each other, from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy; X2 is OR2, NR2bR2c, S (O) mR2d, R2a is selected from C1-4 alkyl, C1-4 haloalkyl, C3-6 cycloalkyl, C3-6 halocycloalkyl, C2-4 alkenyl, C2-4 haloalkenyl, C2-4 alkynyl , C1-4 alkoxy-C1-4 alkyl, phenyl, heteroaryl, heterocyclyl, phenyl-C1-4 alkyl, heteroaryl-C1-4 alkyl and heterocyclyl-C1-4 alkyl, wherein the ring, in the last 6 radicals mentioned, it can be unsubstituted or it can have 1, 2, 3, 4 substituents that are independently selected from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy, and wherein R2b, R2c are independently selected from hydrogen, C1-4 alkyl, C1-4 haloalkyl, C3-6 cycloalkyl, C3-6 halocycloalkyl, C2-4 alkenyl, C2-4 haloalkenyl, C2-4 alkynyl , C1-4 alkoxy-C1-4 alkyl, C1-4 alkylcarbonyl, C1-4 haloalkylcarbonyl, C1-4 alkylsulfonyl, C1-4 haloalkylsulfonyl, phenyl, phenylcarbonyl, phenylsulfonyl, heteroaryl, heteroarylcarbonyl, heteroarylsulfonyl, heterocyclyl, he tert-cyclocarbonyl, heterocyclylsulfonyl, phenyl-C 1-4 alkyl, heteroaryl-C 1-4 alkyl and heterocyclyl C 1-4 alkyl, wherein the ring, in the last 12 radicals mentioned, may not be substituted or may have 1, 2, 3, 4 or 5 substituents that are independently selected from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy; or R2b and R2c, together with the nitrogen atom to which they are attached, form a saturated or unsaturated 5 or 6 membered heterocycle, which may have another heteroatom that is selected from O, S and N as a ring member atom, and wherein the heterocycle may be unsubstituted or may have 1, 2, 3, 4 or 5 substituents that are independently selected from each other from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy, and wherein R2d is selected from C1-4 alkyl, C1-4 haloalkyl, C3-6 cycloalkyl, C3-6 halocycloalkyl, C2-4 alkenyl, C2-4 haloalkenyl, C2-4 alkynyl, C1 alkoxy -4-C 1-4 alkyl, phenyl, heteroaryl, heterocyclyl, phenyl-C 1-4 alkyl, heteroaryl-C 1-4 alkyl and heterocyclyl-C 1-4 alkyl, wherein the ring, in the last 6 radicals mentioned, may not be substituted or may have 1, 2, 3, 4 or 5 substituents that are independently selected from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy; R1 is hydrogen, CN, C1-10 alkyl, C1-10 haloalkyl, C3-10 cycloalkyl, C3-10 halocycloalkyl, C2-10 alkenyl, C2-10 haloalkenyl, C2-10 alkynyl, C3-10 haloalkyl, ORa, C ( Y) Rb, C (Y) ORc, S (O) 2Rd, NReRf, C (Y) NRgRh, S (O) mNReRf, C (Y) NRiNReRf, phenyl, heteroaryl, heterocyclyl, C1-5-ORa alkylene, alkylene C1-5-CN, phenyl-C1-5 alkyl, heteroaryl-C1-5 alkyl, heterocyclyl-C1-5 alkyl, C3-10 cycloalkyl-C1-5 alkyl, C3-10-C (Y) Rb alkylene, C1 alkylene -5-C (Y) ORc, rent C1-5-NReRf, rent C1-5-C (Y) NRgRh, rent C1-5-S (O) 2Rd, rent C1-5-S (O) mNReRf, rent C1-5-C (Y) NRiNReRf, wherein the last 16 radicals mentioned may be unsubstituted or may have 1, 2, 3, 4 or 5 identical or different Rx or Ry substituents; m is 0, 1, 2; Y is O or S; Ra, Rb, Rc are independently selected from hydrogen, C1-4 alkyl, C1-4 haloalkyl, C3-6 cycloalkyl, C3-6 cycloalkylmethyl, C3-6 halocycloalkyl, C2-4 alkenyl, C2-4 haloalkenyl, C2-4 alkynyl, C1-4 alkoxy-C1-4 alkyl, phenyl, heteroaryl, heterocyclyl, phenyl-C1-4 alkyl, heteroaryl-C1-4 alkyl and heterocyclyl-C1-4 alkyl, wherein the ring, in the latter 6 mentioned radicals, may be unsubstituted or may have 1, 2, 3, 4 substituents which are independently selected from each other from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and haloalkoxy C1-4; Rd is selected from C 1-4 alkyl, C 1-4 haloalkyl, C 3-6 cycloalkyl, C 3-6 cycloalkylmethyl, C 3-6 halocycloalkyl, C 2-4 alkenyl, C 2-4 haloalkenyl, C 2-4 alkynyl, C 1-4 alkoxy C1-4, phenyl, heteroaryl, heterocyclyl, phenyl-C1-4 alkyl, heteroaryl-C1-4 alkyl and heterocyclyl-C1-4 alkyl, wherein the ring, in the last 6 radicals mentioned, may be unsubstituted or may have 1, 2, 3, 4 or 5 substituents that are independently selected from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy; Re, Rf are independently selected from hydrogen, C1-4 alkyl, C1-4 haloalkyl, C3-6 cycloalkyl, C3-6 cycloalkylmethyl, C3-6 halocycloalkyl, C2-4 alkenyl, C2-4 haloalkenyl, C2 alkynyl -4, C1-4 alkoxy-C1-4 alkyl, C1-4 alkylcarbonyl, C1-4 haloalkylcarbonyl, C1-4 alkylsulfonyl, C1-4 haloalkylsulfonyl, phenyl, phenylcarbonyl, phenylsulfonyl, heteroaryl, heteroarylcarbonyl, heteroarylsulfonyl, heterocyclyl, heterocyclylcarynyl, heterocyclyl sulfonyl , phenyl-C 1-4 alkyl, heteroaryl-C 1-4 alkyl and heterocyclyl-C 1-4 alkyl, wherein the ring, in the last 12 radicals mentioned, may be unsubstituted or may have 1, 2, 3, 4 or 5 substituents that are independently selected from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy; or Re and Rf, together with the nitrogen atom to which they are attached, form a saturated or unsaturated 5 or 6 membered heterocycle, which may have another heteroatom that is selected from O, S and N as a ring member atom, and wherein the heterocycle may be unsubstituted or may have 1, 2, 3, 4 or 5 substituents that are independently selected from each other from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy; Rg, Rh are independently selected from hydrogen, C1-4 alkyl, C1-4 haloalkyl, C3-6 cycloalkyl, C3-6 halocycloalkyl, C2-4 alkenyl, C2-4 haloalkenyl, C2-4 alkynyl, C1 alkoxy -4-C 1-4 alkyl, phenyl, heteroaryl, heterocyclyl, phenyl-C 1-4 alkyl, heteroaryl-C 1-4 alkyl and heterocyclyl-C 1-4 alkyl, wherein the ring, in the last 6 radicals mentioned, may not be substituted or may have 1, 2, 3, 4 substituents which are independently selected from each other from halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy; Ri is selected from hydrogen, C1-4 alkyl, C1-4 haloalkyl, C3-6 cycloalkyl, C3-6 cycloalkylmethyl, C3-6 halocycloalkyl, C2-4 alkenyl, C2-4 haloalkenyl, C2-4 alkynyl, C1-4 alkoxy -C 1-4 alkyl, phenyl and phenyl-C 1-4 alkyl, wherein the phenyl ring, in the last 2 radicals mentioned, may be unsubstituted or may have 1, 2, 3, 4 or 5 substituents selected, independently of each other, of halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy and C1-4 haloalkoxy; Rx are independently selected from cyano, nitro, C1-4 alkoxy, C1-4 haloalkoxy, C1-4 alkylthio, C1-4 haloalkyl, C1-4 alkylsulfinyl, C1-C4-haloalkylsulfinyl, C1-4 alkylsulfonyl, haloalkylsulfonyl C1-4, C1-10 alkylcarbonyl, C3-6 cycloalkyl, hete |
| priorityDate | 2009-07-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 24.