http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-066715-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_8e0bf0928b608797b70bbc2b91c7e52e |
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C2602-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C2602-08 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-50 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D277-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C275-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C335-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D263-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N47-32 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C279-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D233-50 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N47-44 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D261-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D317-60 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-78 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-76 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D213-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-00 |
| filingDate | 2008-05-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2009-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-066715-A1 |
| titleOfInvention | AMINOAZOLINE AND UREA DERIVATIVES TO COMBAT ANIMAL PESTS |
| abstract | Use of aminoazoline and urea derivatives to combat animal pests. Also a method for controlling animal pests using these compounds, seeds and an agricultural and veterinary composition comprising said specific compounds and derivatives of azoline and urea. Claim 1: The use of compounds of the formula (1) or of one of its salts to combat animal pests characterized in that Z is a group of the formulas (2A), (2B) or (2C), n is 0, 1, 2, 3 or 4; m is 1 or 2; it is the site of union with the rest of the molecule; X is S, O or NR5; Y is S, O or NR5a; T is -ORT1, -SRT2, -OC (O) -RT3, -OC (S) -RT4 or -SC- (S) -RT5, RT1, RT2, RT3, RT4 and RT5 are selected from hydrogen, C1- alkyl 6, C2-6 alkenyl or C2-6 alkynyl, where the last three radicals mentioned may carry 1, 2 or 3 RTa substituents; C3-6 cycloalkyl which may carry 1, 2 or 3 RTb substituents; phenyl which can carry 1 2 or 3 RTc substituents; where the phenyl ring can also be fused with another phenyl ring or a saturated, partially unsaturated or aromatic 5 or 6-membered heterocyclic ring containing 1, 2 or 3 heteroatoms selected from O, S and N and optionally 1 or 2 carbonyl groups as ring members, where the fused ring system can carry 1, 2 or 3 RTc substituents; saturated, partially unsaturated or aromatic 5 or 6 membered heterocycle containing 1, 2 or 3 heteroatoms selected from O, S and N and optionally 1 or 2 carbonyl groups as ring members, which may carry 1, 2 or 3 RTd substituents; or RT3, RT4, RT5 are NRT31RT32, where RT31 and RT32, independently of each other, are selected from hydrogen, C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl, where the last three groups mentioned may carry 1, 2 or 3 RTa substituents, C3-6 cycloalkyl, which may carry 1, 2 or 3 RTb substituents; aryl and arylC 1-4 alkyl, where the aryl moiety in the last two groups mentioned may carry 1, 2 or 3 RTc substituents; or RT31 and RT32 together with the nitrogen atom to which they are attached form a saturated, partially unsaturated or aromatic heterocyclic of 3, 4, 5 or 6 members containing 1, 2 or 3 heteroatoms selected from O, S and N and optionally 1 or 2 carbonyl groups as ring members, where the heterocyclic ring can carry 1, 2 or 3 RTd substituents; R 1 is selected from the group consisting of hydrogen, cyano, C 1-6 alkyl, C 1-6 haloalkyl, C 2-6 alkenyl, C 1-6 alkynyl, C 1-6 alkoxycarbonyl, C 1-6 alkylcarbonyl, C 2-6 alkenylcarbonyl , C2-6 alkynylcarbonyl; C3-6 cycloalkyl, phenyl, benzyl, phenoxycarbonyl, 5 or 6 membered heteroaryl and 5 or 6 membered hetarylmethyl each of the last six radicals mentioned may not be substituted or may carry any combination of 1, 2, 3, 4 or 5 radicals Rb1; R2a, R2b are selected from the group consisting of hydrogen, formyl, CN, C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl, C1-6 alkylcarbonyl, C2-6 alkenyl-carbonyl, C2-6 alkynyl carbonyl, C1-6 alkoxycarbonyl, C1-6-thiocarbonyl alkyl, C1-6-thiocarbonyl alkoxy, wherein the carbon atoms in the aliphatic radicals of the aforementioned groups can carry any combination of 1, 2 or 3 radicals Ra2, C (O) NRaRb, C (S) NRaRb, (SO2) NRaRb, phenyl, benzoyl, phenoxycarbonyl, benzyl, benzylcarbonyl, benzyloxycarbonyl, a saturated, partially unsaturated or aromatic 5 or 6 membered ring, 5 or 6 membered heterylmethyl, hetarylcarbonyl 5 or 6 members, 5 or 6 membered methylcarbonyl, wherein each of the last ten radicals mentioned may not be substituted or may carry any combination of 1, 2, 3, 4 or 5 Rb2 radicals, and where the ring 5 or 6-membered heteroaromatic in hetarylmethyl, hetarylcarbonyl and hetarylmethylcarbonyl co It has 1, 2, 3 or 4 heteroatoms selected from oxygen, sulfur and nitrogen as ring members, and wherein the 5 or 6 membered heterocyclic ring contains 1, 2 or 3 heteroatoms selected from oxygen, sulfur and nitrogen as ring members ; or R1 together with R2a may be C3-5-diyl which may carry 1, 2, 3, 4 or 5 radicals R21 and where one or two methylene groups of the radical C3-5-diyl reach may be replaced by 1 or 2 heteroatoms non-adjacent or groups containing heteroatoms selected from O, S and NR22; R1 together with R2b can also be a carbonyl group of bridge C (O); R2c and R2d, independently from each other, are selected from hydrogen, formyl, C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl, aryl, arylC 1-4 alkyl, hetaryl, heteroylC 1-4 alkyl, C 1-6 alkylcarbonyl, C 1-6 alkyl thiocarbonyl, C 2-6 alkenylcarbonyl, C 2-6 alkynylcarbonyl, C 1-6 alkoxycarbonyl, C 1-6 alkoxy thiocarbonyl, arylcarbonyl, heteroarylcarbonyl, aryloxycarbonyl and heteroyloxycarbonyl, where aliphatic, aromatic or heteroaromatic moieties in the last 17 radicals mentioned may carry 1, 2, 3, 4 or 5 Rc2 radicals, and where hetaryl is a 5 or 6 membered heteroaromatic ring containing 1, 2, 3 or 4 heteroatoms selected from O, S and N as ring members; R3a, R3b, R3c, R3d, independently of each other, are selected from the group consisting of hydrogen, halogen, cyano, nitro, hydroxy, mercapto, amino, haloalkyl C1-6, alkyl C1-6, alkyl C1-6- amino, di- (C1-6 alkyl) amino, C1-6 alkoxy, wherein the carbon atoms in the last 4 radicals mentioned may not be substituted or may carry any combination of 1, 2 or 3 radicals Ra3, C3- cycloalkyl 6, phenyl or benzyl, each of the last 3 radicals mentioned may not be substituted or may carry any combination of 1, 2, 3, 4 or 5 Rb3 radicals; R4a, R4b, independently of each other, are selected from the group consisting of hydrogen, halogen, C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl, C1-6 haloalkyl, wherein the carbon atoms in these groups they can carry any combination of 1, 2 or 3 radicals Ra4, phenyl, benzyl, 5 or 6 member hetaryl and 5 or 6 member hetarylmethyl, each of the last 4 radicals mentioned may not be substituted or they can carry any combination of 1 2, 3, 4 or 5 radicals Rb4, and wherein the heteroaromatic ring of 5 or 6 members in hetarylmethyl and hetaryl contains 1, 2, 3 or 4 heteroatoms selected from oxygen, sulfur and nitrogen as ring members; or R4a together with R4b can also be = O, = NRc or = CRdRe; or R4a together with R4b can also be C2-5-diyl which may carry 1, 2, 3, 4, 5 or 6 R41 substituents and where one or two methylene groups of the C2-5-diyl alkan radical may be replaced by 1 or 2 non-adjacent heteroatoms or groups containing heteroatoms selected from O, S and NR42; or R2a together with R4a can form a bivalent bridge radical selected from the group consisting of C (O) -C (R24a) (R24b), C (S) -C (R24a) (R24b), CH2-C (R24a) (R24b), S (O) 2-C (R24a) (R24b), S (O) -C (R24a) (R24b), C (O) -O, C (S) -O, S (O) 2 -O, S (O) -O, C (O) -NH, C (S) -NH, S (O) 2-NH, S (O) -NH; R4c, R4d are defined, independently, as R4a and R4b; R5, R5a, independently of each other, are selected from the group consisting of hydrogen, formyl, CN, C1-6 alkyl, C2-6 alkenyl, C2-6 alkynyl, C1-6 alkylcarbonyl, C2-6 alkenyl carbonyl, C2-6 alkynylcarbonyl, C1-6 alkoxycarbonyl, C1-6 alkylthiocarbonyl, wherein the carbon atoms in the aliphatic radicals of the aforementioned groups can carry any combination of 1, 2 or 3 radicals Ra5, C (O) NRaRb, (SO2) NRaRb, C (S) NRaRb, phenyl, benzyl, phenoxycarbonyl, 5 or 6 membered heteroaryl methyl, 5 or 6 membered heteroylcarbonyl and benzoyl each of the last 6 radicals mentioned may not be substituted or they can carry any combination of 1, 2, 3, 4 or 5 Rb5 radicals, and wherein the 5 or 6 membered heteroaromatic ring in hetarylmethyl and hetarylcarbonyl contains 1, 2, 3 or 4 heteroatoms selected from oxygen, sulfur and nitrogen as members From the ring; each Rz1 is independently selected from the group consisting of halogen, OH, SH, SO3H, COOH, cyano, nitro, C1-6 alkyl, C1-6 alkoxy, C1-6-thio alkyl, C2-6 alkenyl, C2-6-oxy alkenyl, C2-6-thio alkenyl, C2-6 alkynyl, C2-6-oxy alkynyl, C2-6-thio alkynyl, C1-6-sulfonyl alkyl, C1-6-sulfoxyl alkyl, C2-alkenyl 6-sulfonyl, C2-6 alkynyl sulfonyl, a NRaRb radical, formyl, C1-6 alkylcarbonyl, C2-6 alkenylcarbonyl, C2-6 alkynylcarbonyl, C1-6 alkoxycarbonyl, C2-6 alkoxycarbonyl, C2-6-oxycarbonyl alkynyl, formyloxy, C1-6-carbonyloxy alkyl, C2-6-alkynyl, C2-6 alkynylcarbonyloxy, wherein the carbon atoms in the aliphatic radicals of the aforementioned groups can raise any combination of 1 2, 3, 4 or 5 radicals Raz, C (O) NRaRb, (SO2) NRaRb, and radicals of the formula L-Cy, where L is a single bond, oxygen, sulfur or C1-6-diyl, where a carbon can be replaced by oxygen, Cy is selected from the group consisting of C3-12 cycloalkyl, which is unsubstituted or which is substituted with any combination of 1, 2, 3, 4 or 5 radicals Rbz, phenyl, naphthyl and 5- or 10-membered mono- or bicyclic heterocyclyl, which it contains 1, 2, 3 or 4 heteroatoms selected from oxygen, sulfur and nitrogen as ring members, where Cy is not substituted or can carry any combination of 1, 2, 3, 4 or 5 Rbz radicals; and wherein two radicals Rz1 that are attached to adjacent carbon atoms can form together with said carbon atoms a fused benzene ring, a fused, saturated or partially unsaturated carbocycle of 5, 6 or 7 members or a fused heterocycle of 5, 6 or 7 members, containing 1, 2, 3 or 4 heteroatoms selected from oxygen, sulfur and nitrogen as ring members, and where the fused ring is not substituted or can carry any combination of 1, 2, 3 or 4 radicals Rbz ; Ra, Rb are selected |
| priorityDate | 2007-05-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 51.