http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-062678-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_173bc2c63b34988699010ba05e5b1376 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-42 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-12 |
| filingDate | 2007-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2008-11-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-062678-A1 |
| titleOfInvention | AMINES OF CHINOLINYLOXIALCANOIC ACID WITH FUNGICIDE PROPERTIES |
| abstract | These compounds are useful as fungicides and bactericides used in agriculture and horticulture. Claim 1: A compound of General Formula (1) wherein Q1, Q2 and Q3, independently of each other, are optionally substituted halogen, cyano, nitro, azido, C1-6 alkyl, optionally substituted cycloalkyl (C3-6), optionally substituted heterocyclyl (C3-6), containing at least one heteroatom selected from sulfur, oxygen or NR0, where R0 is hydrogen or optionally substituted (C1-6) alkyl, (C3-6) cycloalkyl (C1-4) alkyl optionally substituted, optionally substituted (C2-6) alkenyl, optionally substituted alkynyl (C2-6), optionally substituted alkoxy (C1-6), optionally substituted alkenyloxy (C2-6), optionally substituted alkynyloxy (C2-6) alkyloxy, aryl optionally substituted, optionally substituted aryloxy, optionally substituted arylalkyl (C1-6), optionally substituted arylalkoxy, optionally substituted heteroaryl, optionally substituted heteroaryloxy, optionally substituted heteroarylalkyl (C1-6), heteroarylalkyl (C1-6) Nally substituted, -SF5 or -S (O) ual (C1-6) alkyl, where u is 0.1 or 2 and the alkyl group is optionally substituted with halogen, or Q1, q2 and Q3, independently of each other, are - OSO2 (C1-4) alkyl, where the alkyl group is optionally substituted with halogen, or Q1, Q2 and Q3, independently of one another, are -CONRuRv, -CORu, -CO2Ru, -CRu = NRv, -NRuRv, -NRuCORv, - NRuCO2Rv, -SO2NRuRv or -NRuSO2Rw, where Rw is optionally substituted (C1-6) alkyl and Ru and Rv, independently of each other, are hydrogen or (C1-6) alkyl optionally substituted with halogen, or, in the case of -CONRuRv or -SO2NRuRv, RuRv can be joined to form a 5- or 6-membered carbocyclic or heterocyclic ring containing a heteroatom selected from sulfur, oxygen and NR0, where R0 is hydrogen or optionally substituted (C1-6) alkyl, or, in the case of -CRu = NRv, Rv is optionally substituted hydroxy or (C1-6) alkoxy, optionally substituted aryloxy or optionally substituted heteroaryloxy, or Q1 and Q2, independently of each other, further indicate hydrogen, R1 is optionally substituted (C1-4) alkyl, optionally substituted alkenyl (C2-4), optionally substituted alkynyl (C2-4) or optionally substituted cycloalkyl (C3-4) , R2 is hydrogen, (C1-8) alkyl, (C3-4) cycloalkyl, (C2-8) alkenyl, cyano, hydroxy, alkoxy, cyanoalkyl (C1-4), (C1-4) alkoxy (C1-4) alkyl ), (C1-4) alkoxy (C1-4) alkoxy (C1-4) alkyl or benzyloxyalkyl (C1-4), where the phenyl ring is optionally substituted with (C1-4) alkoxy, R3 is - (CRaRb) p (CRcRd) q (X) r (CReRf) sR4, where Ra, Rb, Rc, Rd, Re and Rf, independently of each other, are hydrogen, (C1-4) alkyl, halogen, cyano, hydroxy, (C1) alkoxy -4) or (C1-4) alkoxycarbonyl, or RaRb, RcRd or ReRf can be joined to form a 3- to 8-membered carbocyclic or heterocyclic ring containing a heteroatom selected from sulfur, oxygen and NR0, where R0 is hydrogen or alkyl (C1-6) optionally substituted, X is (CO), (CO) O, O (CO), O, S (O) t, where T is 0, 1 or 2, or X is NH or Nalkyl (C1-6), p, rys, independent of each other, are 0 or 1, which is 0, 1 or 2, R4 is (C1-6) alkyl optionally substituted, optionally substituted (C2-6) alkenyl, -CRuu = NRvv, where Ruu is hydrogen or (C1-6) alkyl and Rvv is hydroxy or optionally substituted (C1-6) alkoxy, optionally substituted aryloxy or optionally substituted heteroaryloxy, or -CH2-C ::: C-R5, where R5 is hydrogen, (C1-8) alkyl optionally substituted with halogen, hydroxy, (C1-6) alkoxy, (C1-3alkoxy (C1-3, cyano, alkyl) (C1-4) carbonyloxy, aminocarbonyloxy, mono- or di- (C1-4) aminocarbonyloxy, trialkyl (C1-4) silyloxy or -S (O) (1-6C) alkyl, where g is 0, 1 or 2 , or R5 is (C3-6) cycloalkyl optionally substituted with halogen, hydroxy, (C1-6) alkoxy, (C1-3) alkoxy (C1-3) alkoxy, cyano, (C1-4carbonyloxy, aminocarbonyloxy, mono- or di- (C1-4) aminocarbonyloxy, trialkyl (C1-4silyloxy or -S (O) (C1-6) alkyl, where g is 0, 1 or 2, or R5 is (C3-6) cycloalkyl (C1-) alkyl 4), where the alkyl and / or cycloalkyl portion is optionally substituted with halogen, hydroxy, C1-6 alkoxy, C1-3 alkoxy (C1-3) alkoxy, cyano, C1-4 alkylcarbonyloxy, aminocarbonyloxy, mono- or di - (C1-4) alkylcarbonyloxy, trialkyl (C1-4) silyloxy or -S (O) (C1-6) alkyl, where g is 0, 1 or 2, or R5 is optionally substituted aryl, aryl (C1-4) alkyl ) optionally substituted, optionally substituted aryloxyalkyl (C1-4), optionally substituted heteroaryl or optionally substituted heteroarylalkyl (C1-4) or optionally substituted heteroaryloxyalkyl (C1-4), or R4 is optionally substituted cycloalkyl (C3-6), cycloalkenyl (C5 -6) optionally substituted, optionally substituted aryl, optionally substituted heteroaryl or an optionally substituted 5 to 8-membered ring optionally containing a heteroatom selected from sulfur, oxygen or NR0, where R0 is hydrogen or optionally substituted (C1-6) alkyl, or when R3 is - (CRaRb) p (CRcRd) q (X) r (CReRf) sR4, R2 and R3 can n to form a 5- or 6-membered ring optionally substituted with halogen, (C1-4) alkyl, mono- or di- (C1-4) aminocarbonyl, which optionally contains a heteroatom selected from sulfur, oxygen and NR0, where R00 is (C1-4) alkyl optionally substituted with halogen, (C1-6) alkoxy or cyano, or R00 is phenyl optionally substituted with nitro, (C1-4) alkyl, halo (C1-4) alkyl, (C1-) alkyl 4) carbonyl or heteroaryl, or R2 and R3 can be joined to form an optionally substituted 6.6-membered bicyclo, R3 is - (CR3R40) C ::: CR50, where R30 and R40, independently of each other, are hydrogen, (C1-6) alkyl, halo (C1-4) alkyl, (C1-4) alkoxy (C1-3) alkyl, (C2-3) alkenyl or (C2-3) alkynyl, or R30 and R40 bond with the atom carbon to which they are attached to form a 3- to 6-membered carbocyclic or heterocyclic ring containing in heteroatom selected from sulfur, oxygen or NR00, where R000 is hydrogen or (C1-4) alkyl, where the carbocyclic ring co or heterocyclic is optionally substituted with halo or (C1-4) alkyl, R50 is hydrogen, optionally substituted (C1-4) alkyl, optionally substituted cycloalkyl (C3-6), optionally substituted aryl or optionally substituted heteroaryl containing a selected heteroatom between sulfur, oxygen or NR000, where R000 is hydrogen or (C1-6) alkyl, L is sulfur or oxygen, and n is 0, 1 or 2, and salts and N-oxides of the compounds of Formula 1. |
| priorityDate | 2006-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 31.