http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-058385-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_981a37900e6991fb373304ed2ba5a703 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N53-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D213-61 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D333-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N47-48 |
| filingDate | 2006-12-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2008-01-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-058385-A1 |
| titleOfInvention | CARBOXAMIDS EMPLOYED IN THE FIGHT AGAINST INDESEABLE MICROORGANISMS, COMPOSITIONS THAT CONTAIN THEM AND METHOD OF OBTAINING THEMSELVES AND A PROCEDURE FOR THE PREPARATION OF THESE CARBOXAMIDS AND INTERMEDIARIES OF SYNTHESIS OF THE SAME. |
| abstract | Several procedures for obtaining these products and their use for the fight against undesirable microorganisms, as well as intermediate products and compositions containing these carboxamides. Claim 1: Carboxamides of the formula (1), wherein X means OR1, SR2. NHR3, NR4R5, SOR8, SO2R6; R1 means C1-12 alkyl, C2-8 alkenyl, C2-8 alkynyl; C1-8 haloalkyl, hydroxy-C1-8 alkyl, (C1-4 alkoxy) -C1-8 alkyl, bis (C1-4 alkoxy) -C1-8 alkyl, (C1-4 alkoxy) carbonyl- (C1-4 alkyl ); phenyl- (C1-2 alkyl) or heteroaryl- (C1-2 alkyl) respectively, if necessary, substituted by halogen, C1-4 alkyl or C1-4 haloalkyl; (C1-6 alkyl) carbonyl, (C3-8 cycloalkyl) carbonyl, phenylcarbonyl or hetarylcarbonyl substituted respectively, where appropriate, by C1-4 alkoxy, by halogen, by C1-4 alkyl or by C1-4 haloalkyl; R 2 means C 1-12 alkyl, C 2-8 alkenyl, C 2-8 alkynyl, C 1-8 haloalkyl, C 1-8 hydroxy-alkyl, (C 1-4 alkoxy) -C 1-8 alkyl, bis (C 1-4 alkoxy) -alkyl C1-8, cyano- (C1-4 alkyl), -OH2S-CN, (C1-4 alkoxy) -carbonyl- (C1-4 alkyl); phenyl- (C1-2 alkyl) or heteroaryl- (C1-2 alkyl) substituted respectively, where appropriate, by halogen, by C1-4 alkyl or by C1-4 haloalkyl; (C1-6 alkyl) carbonyl, (C3-8 cycloalkyl) carbonyl, phenylcarbonyl or hetarylcarbonyl substituted respectively, where appropriate, by C1-4 alkoxy, halogen: C1-4 alkyl or C1-4 haloalkyl; R3, R4 and R5 mean, independently of each other, amino, hydroxyl, cyano, C1-12 alkyl, C1-8 alkoxy, C2-8 alkenyl, C2-8 alkynyl, C1-6 alkylamino, di (C1-6 alkyl) amino , hydroxy-C 1-8 alkyl, (C 1-4 alkoxy) -C 1-8 alkyl, bis (C 1-4 alkoxy) -C 1-8 alkyl, cyano- (C 1-4 alkyl), phenoxy, phenylamino, benzyloxy or benzylamino; R6 means C1-12 alkyl or C1-8 haloalkyl; M means a phenyl, thiophene, pyridine, pyrimidine, pyridazine or substituted pyrazine ring, respectively, once by R7 or means a thiazole ring substituted by R8; R7 means hydrogen, fluorine, chlorine, methyl, isopropyl, methylthio or trifluoromethyl; R8 means hydrogen, methyl, methylthio or trifluoromethyl; Q means a direct bond, C1-4 alkylene, C2-4 alkenylene, O, S, SO, SO2 or NR9; R9 hydrogen, C1-8 alkyl, C1-4 alkoxy- C1-4 alkyl, C1-4 alkylthio-C1-4 alkyl, C2-8 alkenyl, C2-8 alkynyl, C1-6 haloalkyl, C2-6 haloalkenyl, C2 haloalkynyl -6 or C3-6 cycloalkyl; Z means z1, Z2, Z3, z4, z5 or Z6; Z1 means phenyl substituted, where appropriate, one to five times, by identical or different substituents; z2 means pyridinyl substituted, where appropriate, one to three times, by identical or different substituents; Z3 means cycloalkyl or bicycloalkyl substituted respectively, where appropriate, once or several times, by identical or different substituents, such as by halogen, by alkyl and / or by (CR10R11) mSiR12R13R14; z4 means unsubstituted C2-20 alkyl or means C1-20 alkyl substituted once or several times, by identical or different substituents, by halogen, by alkylthio, by alkylsulfinyl, by alkylsulfonyl, by alkoxy, by alkylamino, by dialkylamino, by haloalkylthio, by haloalkylsulfinyl, by haloalkylsulfonyl, by haloalkoxy, by haloalkylamino, by halodialkylamino, by -SiR12R13R14 and / or by C3-6 cycloalkyl, the cycloalkyl part may be substituted, if appropriate, once or several times, by identical substituents or different, by halogen and / or C1-4 alkyl; Z5 means C2-20 alkenyl or C2-20 alkynyl substituted respectively, where appropriate, once or several times, by identical or different substituents, by halogen, by alkylthio, by alkylsulfinyl, by alkylsulfonyl, by alkoxy, by alkylamino, by dialkylamino, by haloalkylthio, by haloalkylsulfinyl, by haloalkylsulfonyl, by haloalkoxy, by haloalkylamino, by halodialkylamino, by -SiR12R13R14 and / or by C3-6 cycloalkyl, the cycloalkyl part may be substituted, if appropriate, once or several times, by identical or different substituents such as halogen and / or C1-4 alkyl; Z6 means a ring with 3 to 7 members, saturated or unsaturated, substituted, where appropriate, once or several times, containing a silicon atom as a member of the ring, then Q meaning a direct bond or C1-4 alkylene; R10 means hydrogen or C1-4 alkyl; R11 means hydrogen or C1-4 alkyl; m means 0, 1, 2 or 3; R12 and R13 mean, independently of each other, hydrogen, C1-8 alkyl, C1-8 alkoxy, C1-4 alkoxy-C1-4 alkyl, C1-4 alkylthio-C1-4 alkyl or C1-6 haloalkyl; R14 means hydrogen, C1-8 alkyl, C1-8 alkoxy, C1-4 alkoxy-C1-4 alkyl, C1-4 alkylthio-C1-4 alkyl, C2-8 alkenyl, C2-8 alkynyl, C1-6 haloalkyl, haloalkenyl C2-6, C2-6 haloalkynyl, C3-6 cycloalkyl, or means substituted phenyl or phenylalkyl respectively, if appropriate, or MQZ together, mean, 1H-2,3-dihydroinden-4-yl, 1,3-dihydro -2-benzofuran-4-yl or 1,3-dihydro-2-benzothien-4-yl substituted respectively, where appropriate, one to three times per methyl; A means one of the radicals A1 through A19 of the group of formulas (2); R15 means hydrogen, cyano, halogen, nitro, C1-4 alkyl, C1-4 alkoxy, C1-4 alkylthio, C3-6 cycloalkyl, C1-4 haloalkyl, C1-4 haloalkoxy or C1-4 haloalkyl with, respectively, 1 to 5 halogen, aminocarbonyl or aminocarbonyl-C1-4 alkyl atoms; R16 means hydrogen, halogen, cyano, C1-4 alkyl, C1-4 alkoxy or C1-4 alkylthio; R17 means hydrogen, C 1-4 alkyl, hydroxy-C 1-4 alkyl, C 2-6 alkenyl, C 3-6 cycloalkyl, C 1-4 alkylthio-C 1-4 alkyl, C 1-4 alkoxy-C 1-4 alkyl, C 1-4 haloalkyl , C1-4 haloalkyl C1-4alkyl, C1-4 haloalkoxy-C1-4alkyl with, respectively, 1 to 5 halogen or phenyl atoms; R18 and R19 mean, independently of each other, hydrogen, halogen, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R20 means halogen, cyano or C1-4 alkyl, or C1-4 haloalkyl or C1-4 haloalkoxy with, respectively, 1 to 5 halogen atoms; R21 and R22 mean, independently of each other, hydrogen, halogen, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R23 means hydrogen, halogen, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R24 means hydrogen, halogen, hydroxy, cyano, C 1-6 alkyl, C 1-4 haloalkyl, C 1-4 haloalkoxy or C 1-4 haloalkyl with, respectively, 1 to 5 halogen atoms; R25 means halogen, hydroxy, cyano, C 1-4 alkyl, C 1-4 alkoxy, C 1-4 alkylthio, C 1-4 haloalkyl, C 1-4 haloalkyl or C 1-4 haloalkoxy with, respectively, 1 to 5 halogen atoms; R26 means hydrogen, halogen, cyano, C1-4 alkyl, C1-4 alkoxy ,. C 1-4 alkylthio, C 1-4 haloalkyl, C 1-4 haloalkoxy with, respectively, 1 to 5 halogen atoms, C 1-4 alkylsulfinyl or C 1-4 alkylsulfonyl; R27 means C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R28 means C1-4 alkyl; Q1 means S (sulfur), SO, SO2 or CH2; p means 0, 1 or 2, R28 being identical or different radicals, when p means 2; R29 means C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R30 means C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R31 and R32 mean, independently of each other, hydrogen, halogen, amino, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R33 means hydrogen, halogen, C1-4 alkyl or C1-4 haloalkyl, with 1 to 5 halogen atoms; R34 and R35 mean, independently of each other, hydrogen, halogen, amino, nitro, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R36 means hydrogen, halogen, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R37 means hydrogen, halogen, amino, C1-4 alkylamino, di- (C1-4 alkyl) amino, cyano, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R38 means halogen, C1-4 alkyl C1-4 haloalkyl, with 1 to 5 halogen atoms; R39 means hydrogen, halogen, amino, C1-4 alkylamino, di- (C1-4 alkyl) amino, cyano, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R40 means halogen, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R41 means halogen, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R42 means hydrogen or C1-4 alkyl; R43 means halogen or C1-4 alkyl; R44 means C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R45 means hydrogen, halogen, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R46 means halogen, hydroxy, C1-4 alkyl, C1-4 alkoxy, C1-4 alkylthio, C1-4 haloalkyl, C1-4 haloalkyl or C1-4 haloalkoxy with, respectively, 1 to 5 halogen atoms; R47 means hydrogen, cyano, C1-4 alkyl, C1-4 haloalkyl with 1 to 5 halogen atoms, C1-4 alkoxy-C1-4 alkyl, hydroxy-C1-4 alkyl, C1-4 alkylsulfonyl, di (C1- alkyl 4) aminosulfonyl, C1-6 alkylcarbonyl or substituted phenylsulfonyl or benzoyl respectively, if appropriate; R48 means hydrogen, halogen, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R49 means hydrogen, halogen, cyano, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R50 means hydrogen, halogen, C1-4 alkyl or C1-4 haloalkyl with 1 to 5 halogen atoms; R51 means C1-4 alkyl. |
| priorityDate | 2005-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 53.