http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-055606-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_cf32b60391b469c41e86c353437f5751 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D239-74 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D265-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D217-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D239-70 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D217-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-12 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D217-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D217-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D239-70 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-06 |
| filingDate | 2006-08-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2007-08-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-055606-A1 |
| titleOfInvention | BENZOQUINAZOLINE DERIVATIVES |
| abstract | Pharmaceutical composition, process and use to prevent or treat bone conditions. Claim 1: A compound of the formula (1) or a pharmaceutically acceptable salt or prodrug ester thereof, wherein: Q is CH or N; R2 is C1-4 alkyl; Y is selected from the group consisting of R5-O-, C1-4 alkyl, C1-4 alkenyl, C1-4 alkynyl, R5-NH-; wherein R5 is C1-4 alkyl, C1-4 alkenyl, C1-4 alkynyl; X is selected from the group consisting of aryl, heteroaryl, C1-10 alkyl, C1-10 alkyloxy, cycloalkyl, heterocycle-alkyl, aryl-C1-4 alkyl, heteroaryl-C1-4 alkyl, cycloalkyl-C1 alkyl -4, heterocycloalkylC 1-4 alkyl, aryl amino, heteroaryl amino, arylC 1-4 alkyl, heteroarylC 1-4 alkyl, C 1-6 alkyl, C 1-6 amino dialkyl, aryloxy, heteroaryloxy, arylC 1-4 alkyloxy, heteroarylC 1-4 alkyloxy, cycloalkylC 1-4 alkyl, heterocycloalkylC 1-4 alkyl-amino, cycloalkylC 1-4 alkyloxy, or heterocyclo-alkylC 1-6 alkyloxy -4, each of which is optionally substituted one or more times; the substituent or optional substituents on X being selected independently from the group consisting of halogen, cyano, trifluoro-methyl, nitro, hydroxyl, (C1-4 alkyl, C1-4 alkyloxy, amino, sulfanyl, sulfonyl, amino, oxycarbonyl, hydroxy, sulfinyl, amino-sulfonyl, sulfonyl-amino, carbonyl, carbonyloxy, carbonyl-amino, carboxyl, acyl, acylamino, or carbamoyl) optionally substituted; the substituent or optional substituents being selected from C1-6 alkyl, C1-6 alkyloxy, carboxyl, hydroxyl, hydroxy-C1-4 alkyl, each of which in turn may be optionally substituted by C1-6 alkyloxy, alkyl C1-6, fluorinated C1-3 alkyl, C1-6 alkyloxy, carboxyl, hydroxyl, hydroxy-C1-4 alkyl, halogen, cyano, nitro; R3 and R4 each represents one or more substituents independently selected from: H, halogen, C1-4 alkyl, C1-4 alkyloxy, CF3; the substituent or optional substituents being selected on R 3 or R 4 independently from the group consisting of C 1-4 alkyl, halogen, C 1-4 alkyloxy, cyano, sulfanyl, sulfonyl, amino, oxycarbonyl, hydroxyl, which in turn may be optionally substituted one or more times by C1-4 alkyl, halogen, C1-4 alkyloxy, cyano, sulfanyl, sulfonyl, amino, oxycarbonyl, or hydroxyl. |
| priorityDate | 2005-08-15-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 51.