http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-054964-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_fdb2b95ca7f4d374a06f2273bb1677b1 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P21-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P21-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-675 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-65031 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-24 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-2433 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P27-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-6506 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-653 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07F9-2437 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-02 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F9-653 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F9-6506 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F9-6503 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F9-24 |
| filingDate | 2003-12-22-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c0ee4d9cf62b273108b0f7bfc2967f75 |
| publicationDate | 2007-08-01-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-054964-A1 |
| titleOfInvention | A COMPOUND THAT INCLUDES PHOSPHORAMIDE DERIVATIVES, PROCEDURE TO PREPARE SUCH COMPOUND AND ITS USES |
| abstract | Claim 1: A compound comprising derivatives ix phosphoramide characterized by the general formula 1: wherein: each R1 independently represents hydrogen, C1-6 alkyl, C1-6 haloalkyl, phenyl, heteroaryl or phenyl C1-3 alkyl, wherein all the rings of phenyl and heteroaryl may be optionally substituted by one or more halogen, C1-4 alkyl or C1-4 alkoxy groups, or the two R1 substituents may be attached by completing a saturated or partially unsaturated 5 or 6 membered ring, which may optionally be fused to a benzene ring; A represents an unsaturated or partially unsaturated 5 or 6-membered ring that may optionally contain 1 to 3 heteroatoms selected from N, O and S, where the two substituents L and D are located on adjacent atoms of ring A, and where A it may also be optionally substituted by one or more R2 substituents; L represents a single bond, -O-, -S- or -NR3-; B represents C1-6 alkyl or a ring selected from phenyl, heteroaryl and C3-7 cycloalkyl, wherein said rings may be optionally substituted by one or more R4 substituents; D represents phenyl or pyridine optionally substituted by one or more halogens; groups A and -SO2NHP (O) (OR1) 2 are located on the D-ring available for each other; Each R2 independently represents halogen, cyano, nitro, carboxy, C1-4 alkyl, C2-4 alkenyl, C2-4 alkynyl, C1-4 haloalkyl, hydroxy, C1-4 hydroxyalkyl, C1-4 alkoxy, C1-4 haloalkoxy, C1 -4 alkylthio, amino, C1-4 alkylamino, C1-4 dialkylamino, formyl, C1-4 alkylcarbonyl, C1-4 alkoxycarbonyl, C1-4 haloalkoxycarbonyl, C1-4 alkoxy-C1-3 alkyl, C1-4 alkylcarbonyloxy-C1- 3 alkyl, C3-7 cycloalkyl-C1-4 alkoxy-C1-3 alkyl or C3-7 cycloalkoxy-C1-3 alkyl, or 2 R2 substituents on the same carbon atom can together form an oxo group; R3 represents hydrogen or C1-4 alkyl; Each R4 independently represents halogen, cyano, nitro, carboxy, C1-4 alkyl, C1-4 haloalkyl, hydroxy, C1-4 hydroxyalkyl, C1-4 alkoxy, C1-4 haloalkoxy, C1-4 alkylthio, amino, C1-4 alkylamino , C1-4 dialkylamino, formyl, C1-4 alkylcarbonyl, C1-4 alkoxycarbonyl or C1-4 haloalkoxycarbonyl, or 2 R4 substituents on the same carbon atom may together form an oxo group, and additionally one of the R4 substituents may represent a 5 or 6-membered ring, saturated, unsaturated or partially unsaturated which may optionally contain 1 to 3 heteroatoms selected from N, O and S and which may be optionally substituted by one or more R5 substituents; each R5 independently represents halogen, hydroxy, nitro, cyano, amino, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 alkylcarbonyl, or 2 R5 substituents on the same carbon atom can together form a group oxo; and heteroaryl in the above definitions represents pyridine, pyrazine, pyrimidine or pyridazine; and its salts and solvates. |
| priorityDate | 2002-12-24-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 55.