http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-050630-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_ae84948901b77f34fd51c41264d8d19c |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D473-40 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D473-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-02 |
| filingDate | 2005-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9a206088242d6c969bedd3a0af34b727 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8ead580b442c40b68770298cd0ffe3c9 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_77ad62a7c27c8327b1465e5442adc446 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c3a4a8c06b0135392be6f6cb0075a0e5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c7cf3ded0ef7bdace0069783ffea7aa2 |
| publicationDate | 2006-11-08-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-050630-A1 |
| titleOfInvention | DERIVATIVES OF 6- TRIFLUOROMETIL PURINA 2- REPLACED WITH ANTAGONIST ACTIVITY OF ADENOSINA-A3. PROCESSES OF OBTAINING AND PHARMACEUTICAL COMPOSITIONS. |
| abstract | This is about 2-substituted 6-trifluoromethyl purine derivatives with adenosine-A3 antagonist activity, production processes and pharmaceutical compositions. Claim 1: Compounds of the general formula (1) wherein: R1 represents - [X- (CH2) n] mY, in which formula X is NH or O, n is 0, 1, 2 or 3, m is 0 or 1, and Y is an optionally substituted 5 or 6-membered aromatic or non-aromatic ring, containing 0, 1 or 2 heteroatoms selected from N, O and S, or R 1 represents a nitro group; R2 is H, C1-3 alkyl, ribose, -CH2-O-CO-O-t-butyl or aryl- (C1-3) alkyl; R3 represents H, halogen, NH2, -NH- (C1-6) alkyl, -N-di (C1-6) alkyl, -NH-cycle (C3-8) alkyl, C2-4-alkenyl (hetero) aryl or C2-4-alkynyl (hetero) aryl, from which the heteroatoms are selected from N, O and S, and whose (hetero) aryl groups may be optionally substituted, or R3 represents a 5- or 6-membered aromatic or non-aromatic ring , optionally substituted, containing 0, 1 or 2 heteroatoms selected from N, O and S, and tautomers, stereoisomers and salts thereof. |
| priorityDate | 2004-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 22.