http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-047527-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_227dd812f56cc52ac96b934923e1e2bf |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D333-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D333-28 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D495-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-40 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D307-68 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-08 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D307-68 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D495-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-40 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D333-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-10 |
| filingDate | 2005-02-01-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2006-01-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-047527-A1 |
| titleOfInvention | 2-HALOGENOFURIL / TIENIL-3-CARBOXAMIDAS |
| abstract | Its use for the fight against unwanted microorganisms, as well as new intermediate products and their obtaining. Claim 1: 2-halogenofuryl / thienyl-3-carboxamides of the formula (1), wherein: A means O (oxygen) or S (sulfur); Hal means halogen; R means hydrogen, C 1-8 alkyl, C 1-6 alkylsulfinyl, C 1-6 alkylsulfonyl, (C 1-4) alkoxy-C 1-4 alkyl, C 3-8 cycloalkyl; C1-6 halogenoalkyl, C1-4 halogenoalkylthio, C1-4 halogenoalkylsulfinyl, C1-4 halogenoalkylsulfonyl, halogen (C1-4) -alkoxy (C1-4), halogen C3-8 alkyl with, respectively, 1 to 9 fluorine atoms , of chlorine and / or bromine; formyl, formyl (C1-3) alkyl, (C1-3 alkyl) carbonyl (C1-3) alkyl, (C1-3 alkoxy) carbonyl (C1-3) alkyl; halogen- (C1-3 alkyl) carbonyl (C1-3 alkyl), halogen- (C1-3 alkoxy) carbonyl (C1-3) alkyl with, respectively, 1 to 13 fluorine, chlorine and / or bromine; (C 1-8 alkyl), carbonyl, (C 1-8 alkoxy) carbonyl, (C 1-4 alkoxy) -C 1-4 alkyl) carbonyl, (C 3-8 cycloalkyl) carbonyl; (C1-6 halogenoalkyl) carbonyl, (C1-6 halogenoalkoxy) carbonyl, (halogen (C1-4) alkoxy (C1-4) alkyl) carbonyl, (halogen C3-8cycloalkyl) carbonyl with, respectively, 1 to 9 atoms fluorine, chlorine and / or bromine; or -C (= O) C (= O) R1, -CONR2R3 or -CH2NR4R5; R 1 means hydrogen, C 1-8 alkyl, C 1-8 alkoxy, C 1-4 alkoxy-C 1-4 alkyl, C 3-8 cycloalkyl; C1-6 halogenoalkyl, C1-6 halogenoalkoxy, halogen (C1-4) alkoxy (C1-4) alkyl, halogenocycloalkyl (3-8) with, respectively, 1 to 9 fluorine, chlorine and / or bromine atoms; R2 and R3 mean, independently of each other, respectively, hydrogen, C1-8 alkyl, (C1-4) alkoxy-(C1-4) alkyl, C3-8 cycloalkyl; C1-8 halogenoalkyl, halogen (C1-4) alkoxy (C1-4) alkyl, C3-8 halocycloalkyl, with, respectively, 1 to 9 fluorine, chlorine and / or bromine atoms; R2 and R3 also form, together with the nitrogen atom, with which they are linked, a saturated heterocycle with 5 to 8 atoms in the substituted ring, if given once or several times, equally or in different ways by halogen or by C1-4alkyl, the heterocycle 1 or 2, but not contiguous, heteroatoms of the series consisting of oxygen, sulfur or NR6 may contain; R4 and R5 mean, independently of each other, hydrogen, C1-8 alkyl, C3-8 cycloalkyl; C1-8 halogenoalkyl, C3-8 halogenocycloalkyl, with, respectively, 1 to 9 fluorine, chlorine and / or bromine atoms; R4 and R5 also form, together with the nitrogen atom, with which they are linked, a saturated heterocycle, with 5 to 8 atoms in the substituted ring, if one or several times, equally or in different ways by halogen or C1-4alkyl, the heterocycle 1 or 2 may contain more, non-contiguous heteroatoms, of the series formed or oxygen, sulfur or NR6; R6 means hydrogen or C1-6 alkyl; means a phenyl, thiophene, pyridine, pyrimidine, pyridazine or pyrazine ring monosubstituted, respectively, by R7 or means a thiazole ring substituted by R7-A; R7 means hydrogen, fluorine, chlorine, methyl, iso-propyl, methylthio or trifluoromethyl; R7-A means hydrogen, methyl, methylthio or trifluoromethyl; Z means Z1, Z2, Z3 or Z4, where Z1 means phenyl substituted, where appropriate, one to five times, in the same way or in different ways; Z2 means cycloalkyl or bicycloalkyl substituted respectively, where appropriate, once or several times, in the same way or in different ways; Z3 means unsubstituted C2-20 alkyl or means C1-20 alkyl substituted once or several times, in the same or different ways by halogen, by alkylthio, by alkylsulfinyl, by alkylsulfonyl, by alkoxy, by alkylamino, by dialkylamino, by halogenoalkylthio, by halogenoalkylsulfinyl, by halogenoalkylsulfonyl, by halogenoalkoxy, by halogenoalkylamino, by halogeno-dialkylamino, by -SiR8R9R10 and / or by C3-6 cycloalkyl, the cycloalkyl part may be substituted, for its part, if appropriate, once or several times the same or in different ways by halogen and / or by C1-4 alkyl; Z4 means C2-20 alkenyl or C2-20 alkynyl, substituted respectively, where appropriate, once or several times, in the same way or in different ways by halogen, by alkylthio, by alkylsulfinyl, by alkylsulfonyl, by alkoxy, by alkylamino, by dialkylamino, by halogenoalkylthio, by halogenoalkylsulfinyl, by halogenoalkylsulfonyl, by halogenoalkoxy, by halogenoalkylamino, by halogeno-dialkylamino, by -SiR8R9R10, and / or by C3-6 cycloalkyl, the cycloalkyl part may be substituted, if any, once or several times, in the same way or in different ways by halogen and / or by C1-4 alkyl; R8 and R9 mean, independently of each other, hydrogen, C1-8 alkyl, C1-8 alkoxy, (C1-4) alkoxy-(C1-4) alkyl, (C1-4) alkylthio-(C1-4) alkyl or halogenoalkyl C1-6; R 10 means hydrogen, C 1-8 alkyl, C 1-8 alkoxy, C 1-4 alkoxy-C 1-4 alkyl, C 1-4 alkylthio (C 1-4 alkyl), C 2-8 alkenyl, C 2- alkynyl 8, C1-6 halogenoalkyl, C2-6 halogenoalkenyl, C2-6 halogenoalkynyl, C3-6 cycloalkyl or means substituted phenyl or phenylalkyl respectively, if appropriate; or M and Z together mean 1H-2,3-dihydro-inden-4-yl, 1,3-dihydro-2-benzofuran-4-yl or 1,3-dihydro-2-benzothien-4-yl respectively, if necessary, one to three times per methyl. |
| priorityDate | 2004-02-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 56.