http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-046788-A1
Outgoing Links
Predicate | Object |
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assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_42e94091a4fc81b8d0237117707cc7ee |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D491-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D249-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P11-06 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-52 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-535 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D491-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D209-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-517 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-495 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-50 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D213-64 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D239-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D249-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D317-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D285-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-55 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D221-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D265-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D263-58 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D498-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-54 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D243-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D239-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-14 |
filingDate | 2004-12-03-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c06467c21c093a27397c42d2be4ed5d4 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9e05ebe4974d8da197cf87f789fa5997 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_67071a1e61ab6970f9abc19023cabd7a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e78805a643c89cb7eec63d9a0d1e3010 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_89c388411796e526c64bd9eceea462c9 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5353299f265f73c50a8245a056b7a922 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e49c8a1473bbc3dacafad6a23feb9778 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1040112f8e23489745734a7fc2f2df86 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_aeb10a7418627deb460f7684e72fd2a1 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9ff1c366b4564326966a28e5bb69772c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1b6b0b1940844b58b18e5b4b0b1a688c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fcf8e437843e0467fb8f282154c94497 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7537e14e349cd399e294f25b70790890 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_dc03c445dc231e54d77252342e10e4f2 |
publicationDate | 2005-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | AR-046788-A1 |
titleOfInvention | ANTIGONISTS OF THE PEPTIDE RECEIVER RELATED TO THE CALCITONINE GENE |
abstract | Compounds of formula (1) as antagonists of the peptide receptors related to the calcitonin gene (`` CGRP receptor ''), pharmaceutical compositions comprising them, methods for their identification, methods of treatment with their use, and their use in therapy for the treatment of neurogenic vasodilation, neurogenic inflammation, migraine and other headaches, thermal injury, circulatory shock, suffocations associated with menopause, inflammatory airway diseases, such as asthma and chronic obstructive pulmonary disease (COPD) and others conditions, the treatment of which can be effected by the antagonism of CGRP receptors. Claim 1: A compound characterized in that they are selected from the group consisting of: (ñ) -3- (3-cyano-1H-indole-5-yl) -2 - {[4- (2-oxo) methyl ester -1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carbonyl] -amino} -propionic; [2- [1,4 '] bipiperidinyl-1'-yl-1- (3-cyano-1H-indole-5-yl-methyl) -2-oxo-ethyl] -amide (ñ) -4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; [2- [1,4 '] Bipiperidinyl-1'-yl-1 (3-cyano-7-methyl-1 H -indol-5-yl-methyl) -2-oxo-ethyl] -amide acid (ñ) -4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidine-1-carboxylic acid; (ñ) -3- (7-isopropyl-1H-indazol-5-yl) -2 - {[4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) methyl ester -piperidin-1-carbonyl] -amino} -propionic; [2- [1,4 '] Bipiperidinyl-1'-yl-1 (7-isopropyl-1H-indazol-5-yl-methyl) -2-oxo-ethyl] -amide (ñ) -4- ( 2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; [2- [1,4 '] bipiperidinyl-1'-yl-1 (7-ethyl-1H-indazol-5-yl-methyl) -2-oxo-ethyl] -amide (ñ) -4- ( 2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; [2- [1,4 '] bipiperidinyl-1'-yl-1 (7-methyl-1H-indazol-5-yl-methyl) -2-oxo-ethyl] -amide (ñ) -4- ( 2,2-dioxo-1,4-dihydro-2H-2l6-benzo [1,2,6] thiadiazin-3-yl) -piperidin-1-carboxylic acid; [2- [1,4 '] Bipiperidinyl-1'-yl-1 (7-methyl-3-methyl-1H-indazol-5-yl-methyl) -2-oxo-ethyl] -amide acid (ñ) -4- (2,2-dioxo-1,4-dihydro-2H-2l6-benzo [1,2,6] thiadiazin-3-yl) -piperidin-1-carboxylic acid; (ñ) -2- [4- (6-Cyano-2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carbonyl] -amino] -3- methyl ester (7-methyl-1H-indazol-5- yl) -propionic; {2- [1,4 '] Bipiperidinyl-1'-yl- (7-methyl-1H-indazol-5-yl methyl) -2-oxo-ethyl} -amide (ñ) -4- (6- cyano-2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; {2- [1,4 '] Bipiperidinyl-1'-yl-1- (7-methyl-1H-indazol-5-ylmethyl) -2-oxo-ethyl} -amide acid (ñ) -4- (2 -oxo-1,2,4,5-tetrahydro-benzo [d] [1,3] diazepin-3-yl-1-carboxylic acid; {2- [1,4 '] bipiperidinyl-1'-yl-1- (Ñ) -4- (6-hydroxy-2-oxo- 1,4-dihydro-2H -quinazolin- (7-methyl-1H-indazol-5-yl methyl) -2-oxo-ethyl} -amide 3- il) -piperidin-1-carboxylic acid; {2- [1,4 '] bipiperidinyl-1'-yl-1- (7-methyl-1H-indazol-5-yl methyl) -2-oxo-ethyl} -amide (ñ) -4- (8-methoxy-2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic acid; {2- [1,4 '] bipiperidinyl -1'-yl-1- (7-methyl-1H- indazol-5-ylmethyl) -2-oxo-ethyl} -amide (ñ) -4- (8-chloro-2-oxo-1,4 -dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; (ñ) -N- (3- (7-ethyl-3-methyl-1 H-indazol-5-yl) -1-oxo- 1- (4- (piperidin-1-yl) piperidin- 1-yl) propan-2-yl) -2 ', 3'-dihydro-2'-oxospiro- (piperidin-4,4'-quinazolin) -1 -carboxamide; (ñ) -N- (3- (7-ethyl-3-methyl-1H-indazol-5-yl) -1-oxo-1- (4- (piperidin-1-yl) piperidin-1- il) propan-2-yl) -2,4-dihydro-2'-oxospiro- (piper idin-4,4'-1H-benzo [d] [1,3] oxazin) -1-carboxamide; (ñ) -N- (3- (7- ethyl-1H-indazol-5-yl) -1- (6,7-dihydro-1 H -pyrazol [4,3-c] pyridin-5 (4 H) -yl) -1-oxopropan-2-yl) -4- (1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) piperidin-1-carboxamide; (ñ) -N- (3- (7-ethyl-1H-indazol-5-yl) -1- (6,7-dihydro-7,7-dimethyl-1H-pyrazole [4,3-c] pyridin- 5 (4H) -yl) -1-oxopropan-2-yl) -4- (1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) piperidin-1-carboxamide; (ñ) -methyl 2- (4- (8-fluoro-1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) piperidin-1-carboxamide) -3- (7-methyl-1H-indazol- 5- il) propanoate; (ñ) -4- (8-fluoro-1,2-dihydro-2- oxoquinazolin-3 (4H) -yl) -N- (3- (7-methyl-1H-indazol-5-yl) -1- oxo-1- (4- (piperidin-1-yl) piperidin-1-yl) propan-2-yl) piperidin-1-carboxamide; (ñ) -4- (8-fluoro-1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) -N- (3- (7- methyl-1H-indazol-5-yl) -1- oxo-1- (4-phenylpiperazin-1- yl) propan-2-yl) piperidin-1-carboxamide; (ñ) -4- (8-fluoro-1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) -N (1- (4- (4-fluorophenyl) piperazin-1-yl) -3- (7-methyl-1H-indazol-5-yl) -1-oxopropan-2-yl) piperidin-1- carboxamide; (ñ) -4- (8-fluoro-1,2-dihydro-2-oxoquinazolin- 3 (4H) -yl) -N- (1- (4- (2-fluorophenyl) piperazin-1-yl) -3 - (7-methyl-1H-indazol-5-yl) -1-oxopropan-2-yl) piperidin-1-carboxamide; (ñ) -4- (8-fluoro-1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) -N- (3- (7-methyl- 1H-indazol-5-yl) -1- oxo-1- (4-o-tolylpiperazin-1-yl) propan-2- yl) piperidin-1-carboxamide; (ñ) -methyl 2- (4- (8-fluoro-1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) piperidin-1-carboxamide) -3- (7-ethyl-3-methyl- 1H-indazol-5-yl) propanoate; (ñ) -N- (3- (7-ethyl-3-methyl- 1H-indazol-5-yl) -1-oxo-1- (4- (piperidin-1-yl) piperidin-1- yl) propan -2-yl) -4- (8-fluoro-1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) piperidin-1- carboxamide; (R) -N - ((R) -3- (2-oxo-2,3-dihydro-benzooxazol-6-yl) -1-oxo-1- (4-piperidin-1-yl) piperidin-1- il) propan-2- yl) -4- (8-fluoro-1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) piperidin-1-carboxamide; (ñ) -N- (3- (7-methyl-1 H-indazol-5-yl) -1-oxo-1- (4- (piperidin-1-yl) piperidin-1-yl) propan-2- il) -8'-fluoro-2 ', 3'-dihydro-2'-oxospiro- (piperidin-4,4'-quinazolin) -1-carboxamide; (ñ) -4- (8-fluoro-1,2-dihydro-2,4-dioxoquinazolin- 3 (4H) -yl) -N- (3- (7-methyl-1H-indazol-5-yl) - 1-oxo-1- (4- (piperidin-1-yl) piperidin-1-yl) propan-2-yl) piperidin-1-carboxamide; N - ((R) -3- (2- (trifluoromethyl) -1H-benzo [d] imidazol-5-yl) -1-oxo-1- (4- (piperidin-1-yl) piperidin-1-yl ) propan-2-yl) -4- (1,2-dihydro-2- oxoquinazolin-3 (4H) -yl) piperidin-1-carboxamide; N - ((R) -1- (dimethylcarbamoyl) -2- (2- (trifluoromethyl) -1H-benzo [d] imidazol-5-yl) ethyl) -4- (1,2-dihydro-2-oxoquinazolin- 3 (4H) -yl) piperidin-1- carboxamide; (R) -methyl 2- (4- (1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) piperidin-1-carboxamido) -3- (2,3-dihydro-2-oxo-1H- benzo [d] imidazol-6-yl) propanoate; N - ((R) -3- (2,3-dihydro-2-oxo-1H-benzo [d] imidazol-6-yl) -1-oxo-1 (4-piperidin-1-yl) piperidin-1 - il) propan-2-yl) -4- (1,2-dihydro-2-oxoquinazolin-3 (4H) -yl) piperidin-1- carboxamide; N - ((R) -1- (dimethylcarbamoyl) -2- (2,3-dihydro-2-oxo-1H-benzo [d] imidazol-6-yl) ethyl) -4- (1,2-dihydro- 2-oxoquinazolin-3 (4H) -yl) piperidin-1-carboxamide; N - ((R) -3- (2,3-dihydro-2- oxo-1H-benzo [d] imidazol-6-yl) -1-oxo-1 (4-piperidin-1-yl) piperidin-1 - il) propan-2-yl) -4- (2 ', 3'-dihydro-2'-oxospiro (piperidin-4,4' - (1H) - quinazolin) carboxamide; 4- (1,2-dihydro- 2,4-dioxoquinazolin-3 (4H) -yl) -N - ((R) -3- (7-methyl-1H-benzo [d] [1,2,3] triazol- 5-yl) -1- oxo-1- (4- (piperidin-1-yl) piperidin-1-yl) propan-2- yl) piperidin-1-carboxamide; [2- (4-cyclohexyl-piperazin-1-yl) -2-oxo -1- (2-Oxo-2,3-dihydro-benzooxazol-6-ylmethyl) -ethyl] -amide (R) -4- (2-oxo-1,4-dihydro-2H-quinazolin-3- il) -piperidin-1- carboxylic; [2- (4-isopropyl-piperazin-1-yl) -2-oxo-1- (2- oxo-2,3-dihydro-benzooxazol-6-ylmethyl) -ethyl] -amide of (R) -4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic acid; (R) -N - ((R) -3- ( 2-oxo-2,3-dihydro-benzooxazol-6-yl) -1-oxo-1- (4- (piperidin-1-yl) piperidin-1-yl) propan-2-yl) -2,4- dihydro- 2'-oxospiro- (piperidin-4,4'-1H-benzo [d] [1,3] oxazin) -1-carboxamide; (R) -N - ((R) -3- (2-oxo -2,3-dihydro-benzooxazol-6-yl) -1-oxo-1- (4- (cyclohex-1-yl) piperazin-1-yl) prop an-2-yl) -2,4-dihydro-2'- oxospiro- (piperidin-4,4'-1 H- benzo [d] [1,3] oxazin) -1-carboxamide; (R) -N ((R) -3- (2-oxo-2,3-dihydro-benzooxazol-6-yl) -1-oxo-1- (4- (prop-2-yl) piperazin-1- il) propan-2-yl) -2,4-dihydro-2'-oxospiro- (piperidin-4,4'-1H-benzo [d] [1,3] oxazin) -1-carboxamide; (R) - N - ((R) -3- (2-oxo-2,3-dihydro-benzooxazol-6-yl) -1-oxo- 1- (4- (piperidin-1-yl) piperidin-1 -yl) propan-2-yl) -2,4-dihydro-2'-oxospiro- (piperidin-4,4'-1H-quinazolin) -1-carboxamide; (R) -N - ((R) -3- (2-oxo-2,3-dihydro-benzooxazol-6-yl) -1-oxo-1- (4- (cyclohex-1- yl) piperazin-1 -yl) propan-2-yl) -2,4-dihydro-2'-oxospiro- (piperidin-4,4'-1H-quinazolin) -1-carboxamide; (R) -N - ((R) -3- (2-oxo-2,3-dihydro-benzooxazol-6-yl) -1-oxo-1- (4- (prop-2-yl) piperazin-1 -yl) propan-2-yl) -2,4-dihydro-2'-oxospiro- (piperidin-4,4'-1H-quinazolin) -1-carboxamide; [2- [1,4 '] Bipiperidinyl-1'-yl-1- (4-chloro-2-oxo-2,3-dihydro-benzooxazol-6-ylmethyl) -2-oxo-ethyl] -amide acid (R) -4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; [2- [1,4 '] Bipiperidinyl-1'-yl-1- (5-chloro-2- oxo-2,3-dihydro-benzooxazol-6- ylmethyl) -2-oxo-ethyl] -amide acid (R) -4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; [2- [1,4 '] Bipiperidinyl-1'-yl-1- (4-bromo-2-oxo-2,3-dihydro-benzooxazol-6-ylmethyl) -2-oxo-ethyl] -amide acid (R) -4- (2-Oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; [2- [1,4 '] Bipiperidinyl-1'-yl-1- (5-bromo-2-oxo-2,3-dihydro-benzooxazol-6-ylmethyl) -2-oxo-ethyl] -amide acid (R) -4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; [2- [1,4 '] Bipiperidinyl-1'-yl-1- (4-iodo-2-oxo-2,3-dihydro-benzooxazol-6-ylmethyl) -2-oxo-ethyl] -amide acid (R) -4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-carboxylic; (ñ) -N- (1-Benzyl-2-hydroxy-ethyl) -2- (7-methyl-1H-indazol-5-ylmethyl) -4- oxo-4- [1 ', 2'-dihydro-2 '- oxospiro- [4H-3', 1-benzoxazin-4, 4'-piperidinyl] -butyramide; (ñ) -N (1-Benzyl-2-hydroxy-ethyl) -2- (7-methyl-1H-indazol-5-ylmethyl) -4-oxo-4- [4- (2-oxo-1,4 -dihydro-2H-quinazolin-3-yl) -piperidin-1-yl] -butyramide; N '- {2- (7-methyl-1H- indazol-5-ylmethyl) -4-oxo-4- [4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin (Ñ) -phenyl-acetic acid -1-yl] -butyryl} -hydrazide; (ñ) -1- [1,4 '] bipiperidinyl-1'-yl-4- [4- (8-fluoro-2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin- 1-yl] -2- (7-methyl-1H-indazol-5-ylmethyl) -butane-1,4-dione; (ñ) -1- [1,4 '] bipiperidinyl-1'-yl-2- (7-methyl-1H-indazol-5-ylmethyl) -4- [2', 3'-dihydro-2'-oxospiro - (piperidin-4,4'-quinazolin] -butane-1,4-dione; (ñ) -1- (4-cyclohexyl-piperazin-1-yl) -2- [2-oxo-2-dihydro-benzooxazole -6-ylmethyl] -4- [4- (2-oxo-1,4-dihydro-2H-quinazolin-3-yl) -piperidin-1-yl] -butane-1,4-dione; (ñ) - 1- [1,4 '] bipiperidinyl-1'-yl-2- (2-oxo-2,3-d |
priorityDate | 2003-12-05-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
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