http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-046760-A1
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| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_173bc2c63b34988699010ba05e5b1376 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-90 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N47-38 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N47-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-90 |
| filingDate | 2004-12-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2005-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-046760-A1 |
| titleOfInvention | DERIVATIVES OF SPIROINDOLINE WITH INSECTICIATED PROPERTIES |
| abstract | An insecticidal compound of formula (1), in which Y is a single bond, C = O, C = S, or S (O) m where m is 0, 1 or 2; R1, R2, R3, R4, R8, A1, A2, A3, A4, B1, B2, B3 and B4 are specified organic groups or salts or N-oxides thereof; compositions that contain them and their use to control insects, mites, nematodes or mollusks. Claim 1: A compound of formula (1); in which Y is a simple bond, C = O, C = S, or S (O) m where m is 0, 1 or 2; R1 is hydrogen, optionally substituted alkyl, optionally substituted alkoxycarbonyl, optionally substituted alkylcarbonyl, aminocarbonyl, optionally substituted alkylaminocarbonyl, optionally substituted dialkylaminocarbonyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted alkoxy, optionally substituted aryloxy, optionally substituted heteroaryloxy, optionally substituted heteroxy cyano, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted cycloalkyl, optionally substituted cycloalkenyl, formyl, optionally substituted heterocyclyl, optionally substituted alkylthio, NO or NR13R14, where R13 and R14 are independently hydrogen, COR15, optionally substituted alkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted heterocyclyl or R13 and R14 together with the N atom to which they are attached they form a group -N = C (R16) -NR17R18; R15 is H; optionally substituted alkyl, optionally substituted alkoxy, optionally substituted aryl, optionally substituted aryloxy, optionally substituted heteroaryl, optionally substituted heteroaryloxy or NR19R20; R16, R17 and R18 are each independently H or lower alkyl; R19 and R20 are independently optionally substituted alkyl, optionally substituted aryl or optionally substituted heteroaryl; R2 and R3 are independently hydrogen, halogen, cyano, optionally substituted alkyl, optionally substituted alkoxy or optionally substituted aryl; each R4 is independently halogen, nitro, cyano, optionally substituted C1-8 alkyl, optionally substituted C2-6 alkenyl, optionally substituted C2-6 alkynyl, optionally substituted alkoxycarbonyl, optionally substituted alkylcarbonyl, optionally substituted alkylaminocarbonyl, optionally substituted cycloalkylaminocarbonyl, C3- 7 optionally substituted, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted heterocyclyl, optionally substituted alkoxy, optionally substituted aryloxy, optionally substituted heteroaryloxy, optionally substituted alkylthio or R21R22N, where R21 and R22 are independently hydrogen, C1-8 alkyl, cycloalkyl C3-7, C3-6 alkenyl, C3-6 alkynyl, C3-7 cycloalkyl-C1-4 alkyl, C2-6 haloalkyl, C1-6 alkoxy-C1-6 alkyl, C1-6 or R21 alkoxycarbonyl together with the N atom to which they are attached form a heterocyclic ring of five, six or seven members that may contain one or two additional heteroatoms selected from O, N or S and that may be optionally substituted with one or two C1-6 alkyl groups, or 2 adjacent R4 groups together with the carbon atoms to which they are attached form a carbocyclic or heterocyclic ring of 4, 5, 6 or 7 members which may be optionally substituted with halogen; n is 0, 1, 2, 3 or 4; R8 is optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted cycloalkyl, optionally substituted aryl, optionally substituted alkoxy, optionally substituted aryloxy, optionally substituted alkoxycarbonyl, optionally substituted alkylcarbonyl or optionally substituted alkenylcarbonyl; A1, A2, A3, A4, B1, B2, B3, and B4 are independently hydrogen, hydrogen, halogen, hydroxy, cyano, optionally substituted C1-8 alkyl, optionally substituted C2-6 alkenyl, optionally substituted C2-6 alkynyl, alkoxycarbonyl optionally substituted, optionally substituted alkylcarbonyl, optionally substituted alkylaminocarbonyl, optionally substituted dialkylaminocarbonyl, optionally substituted C3-7 cycloalkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted heterocyclyl, optionally substituted alkoxy, optionally substituted aryloxy, optionally substituted heteroaryloxy, optionally substituted alkyloxy optionally substituted arylthio or R23R24N, where R23 and R24 are independently hydrogen, C1-8 alkyl, C3-7 cycloalkyl, C3-6 alkenyl, C3-6 alkynyl, C3-7 cycloalkyl, C2-6 haloalkyl , C1-6 alkoxy-C1-6 alkyl, C1-6 alkoxycarbonyl or R23 and R24 together with the att mo of N to which they are attached form a five, six or seven membered heterocyclic ring which may contain one or two additional heteroatoms selected from O, N or S and which may be optionally substituted with one or two C1-6 alkyl groups; or A1 and A2 together are = O; or A3 and A4 together are = O; or B1 and B2 together are = O; or B3 and B4 together are = O; or A1 together with B1 is a link; or A3 together with B3 is a link; or A1 together with A2 form with the carbon to which a three to seven member ring is attached and may be saturated or unsaturated and may contain one or two heteroatoms selected from the group consisting of N, O and S and may be optionally substituted with one or two C1-6 alkyl group; or A1 together with B1 form with the carbon to which a three to seven member ring is attached and may be saturated or unsaturated and may contain one or two heteroatoms selected from the group consisting of N, O and S and may be optionally substituted with one or two C1-6 alkyl group; or B1 together with B2 form with the carbon to which a three to seven member ring is attached and may be saturated or unsaturated and may contain one or two heteroatoms selected from the group consisting of N, O and S and may be optionally substituted with one or two C1-6 alkyl group; or A1 together with A3 form a group -CH2-, -CH = CH- or -CH2CH2; or B1 together with B3 form a group -CH2-, -CH = CH- or -CH2CH2; or salts or N-oxides thereof with the proviso that when B1, B2, B3 and B4 are all H, or A1 and A2 are different from H or both A3 and A4 are different from H. |
| priorityDate | 2003-12-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 24.