http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-046322-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_cf32b60391b469c41e86c353437f5751 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C253-32 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C255-29 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N37-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C255-54 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C255-29 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N37-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C255-54 |
| filingDate | 2004-11-04-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2005-11-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-046322-A1 |
| titleOfInvention | AMIDOACETONITRILE COMPOUNDS, METHODS FOR THEIR PREPARATION AND THEIR INTERMEDIARIES AND THEIR USE IN ANTIPARASITARY COMPOSITIONS. |
| abstract | The active ingredients have pesticidal properties. They are especially suitable for the control of parasites both inside and outside warm-blooded animals. Claim 1: A compound of the formula (1), in which: X means Cl, Br or CF3; Y means a simple bond, O, S, S (O) or S (O) 2; and W means O or S. Claim 15: Process for the preparation of compounds of the formula (1), respectively in free form or in salt form, according to claims 1 to 3, wherein a compound of the formula ( 2), which is known or can be produced analogously to corresponding known compounds, and where Y is a single bond, is reacted with a compound of the formula (3), which is known or can be produced analogously to corresponding known compounds, and wherein X is defined as indicated for formula (1), and Q is a labile group, optionally in the presence of a basic catalyst, and, if desired, a compound of the formula (1 ), in which W is O, obtainable according to the method presented or otherwise, respectively in free form or in salt form, is converted into either a compound of the formula (1), in which W is S, for example, by reaction with P4S10, or in another compound of the formula (1), being separated a mixture of isomers obtainable according to the method presented and isolated the desired isomer and / or a free compound of the formula (1) obtainable according to the presented method is converted into a salt or a salt of a compound of the formula (1) obtainable according to the method presented is converted into the free compound of the formula (1) or another salt. Claim 18: Process for the preparation of compounds of the formula (2), respectively in free form or in salt form, for example, characterized in that a compound of the formula (4) is reacted, which is known or can be prepared analogously to corresponding known compounds, and wherein Y is defined as a single bond, and Q is a labile group, with a compound of the formula (5), which is known and can be prepared from hydroxyacetone, a cyanide and ammonia, and, if desired, a compound of the formula (2) obtainable according to the method presented or otherwise, respectively in free form or in salt form, is converted into another compound of the formula (2) , a mixture of isomers obtainable according to the presented method being separated and isolated the desired isomer and / or a free compound of the formula (2) obtainable according to the presented method is converted into a salt or salt of a compound of the FO Formula (2) obtainable according to the method presented is converted into the free compound of the formula (2) or another salt. |
| priorityDate | 2003-11-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 23.