http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-042254-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_227dd812f56cc52ac96b934923e1e2bf |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P33-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-653 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-713 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-78 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N47-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D231-44 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-653 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-44 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N47-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-78 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-713 |
| filingDate | 2003-12-01-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2005-06-15-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-042254-A1 |
| titleOfInvention | DERIVATIVES OF SULFONYLAMINOPIRAZOL PESTICIDES |
| abstract | 5-substituted sulfonylaminopyrazole derivatives, processes for their preparation, compositions of said compounds and their use for the control of pests such as arthropods (insects and arachnids) and helminths (nematodes). Claim 1: A compound of formula (1) wherein R 1 is (C 1-6) alkyl, halo (C 1-6) alkyl, -CN, -C (S) NH 2, or halogen; W is N, -C-CH3 or -C-halogen; R2 is H, -CH3 or halogen; R3 is halo, (C1-6) alkyl, halo (C1-6) alkyl, halo (C1-6) haloalkoxy, S (O) p-halo (C1-6) alkyl or SF5; R4 is H, (C2-6) alkenyl, (C2-6) haloalkenyl, (C2-6) alkynyl, (C2-6) haloalkynyl, (C3-7) cycloalkyl, -CO2-(C1-6) alkyl, - CO2-C3-7 cycloalkyl, -CO2-C1-4 alkyl-C3-7cycloalkyl, -CO2-C3-6 alkenyl, -CO2-C3-6 alkynyl, -CO2- ( CH2) qR7, -CONR8R9, -CO2- (CH2) qR10, - (CH2) qR7, - (CH2) qR10, -COR9, -COCH2NR8R9, -CO- (CH2) qR7 or -CO- (CH2) qR10; or (C1-6) alkyl unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C1-6) alkoxy, halo (C1-6) alkoxy, (C3-7) cycloalkyl, -S (O ) pR11, -CO2-(C1-6) alkyl, -O (C = O) -alkyl (C1-6), NR8R9, CONR8R9, -SO2NR8R9, -OH, -CN, -NO2, -OR7, -OR10, NR8COR12 and NR8SO2R11; R5 is cycloalkyl (C3-7), alkenyl (C2-6), haloalkenyl (C2-6), R13, R10, R17 or -CH = CH-R15, or is (C1-15) alkyl unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C1-6) alkoxy, haloalkoxy (C1-6), alkenyloxy (C3-6), haloalkenyloxy (C3-6), alkynyloxy (C3-6), haloalkyloxy (C3 -6), cycloalkyl (C3-7), -S (O) pR7, -S (O) pR10, -S (O) pR11, -CN, -NO2, -OH, -COR8, NR8COR12, NR8SO2R11, -CONR8R9 , NR8R9, -OR7, -OR10, R13, R10 and -CO2R8, or a methylene group in the unsubstituted or substituted (C1-6) alkyl is replaced by a group selected from -CO, -O-, -S (O ) p-, -NR8-, -COO-, -OCO-, -CONR8-, -NR8CO-, -C (= NOR8) -, -C (= N-NR8R9) - and -C (= NR8) -, provided that the replacement group is not directly linked to the SO2 group in formula (1); R6 and R11 are each independently (C1-6) alkyl, halo (C1-6) alkyl, (C2-6) alkenyl, C2-6 haloalkenyl, (C2-6) alkynyl, (C2-) alkynyl 6) or cycloalkyl (C3-7); R7 is phenyl unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C1-6) alkyl, halo (C1-6) alkyl, (C1-6) alkoxy, (C1-6) haloalkoxy, - CN, -NO2, -S (O) pR11 and NR9R12; R8 is H, (C1-6) alkyl, halo (C1-6) alkyl, cycloalkyl (C3-7), (C1-4) alkyl-cycloalkyl- (C3-7), - (CH2) qR7 or - (CH2) R10; R9 and R12 are each independently H (C1-6) alkyl, halo (C1-6) alkyl, cycloalkyl (C3-7) or alkyl (C1-4) -cycloalkyl (C3-7); or R8 and R9 together with the attached N atom form a saturated ring of five or six members which optionally contains an additional heteroatom in the ring, selected from O, S and N; the ring is unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C 1-6) alkyl and halo (C 1-6) alkyl; R10 and R20 are each independently heterocyclyl unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C1-4) alkyl, halo (C1-4) alkyl, (C1-4) alkoxy , S (O) pR14, -OH, -OR7 and oxo; R13 is aryl unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C1-6) alkyl, haloalkyl (C1-6), alkoxy (C1-6), haloalkoxy (C1-6), - CN, -NO2, -S (O) pR11, -SF5, NR8R9, -COR11, -COR7, -CONR8R9, -SO2NR8R9, -OH, -OR7, R15, R16, -OR16, -SO3H, alkylideneimino (C1-6 ), -CH = NOR14, -S (O) pR18, -CO2R19 and R20; R14 is (C1-6) alkyl or halo (C1-6) alkyl; R15 is phenyl or naphthyl, both unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C1-6) alkyl, haloalkyl (C1-6) and alkoxy (C1-6); R16 is a heteroaromatic radical selected from the group consisting of pyridyl, pyrimidinyl, pyridazinyl, pyrazinyl, triazinyl, thienyl, thiazolyl, thiadiazolyl, oxazolyl, isoxazolyl, furyl, pyrrolyl, pyrazolyl, imidazolyl and triazolyl, wherein said groups are unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C1-6) alkyl, halo (C1-6) alkyl and (C1-6) alkoxy; R17 is a heteroaromatic radical selected from the group consisting of pyridyl, pyrimidinyl, pyridazinyl, pyrazinyl, triazinyl, thienyl, thiazolyl, thiadiazolyl, oxazolyl, isoxazolyl, furyl, pyrrolyl, pyrazolyl, imidazolyl and triazolyl, wherein said groups are unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C1-6) alkyl, halo (C1-6) alkyl and (C1-6) alkoxy; and wherein said heteroaromatic radical is substituted with R15, R16 or -OR16; R18 is phenyl unsubstituted or substituted with one or more radicals selected from the group consisting of halogen, (C1-6) alkyl, haloalkyl (C1-6) and alkoxy (C1-6); R19 is (C1-6) alkyl, halo (C1-6) alkyl, R18 or (C1-6) alkyl (C1-3) alkoxy; n, p and q are, each independently, zero, one or two; and each heterocyclyl in the aforementioned radicals is independently a heterocyclic radical having 3 to 6 ring atoms, and 1, 2, or 3 heteroatoms in the ring selected from the group consisting of N, O and S; or a salt of said compound, acceptable for pesticide use. |
| priorityDate | 2002-12-03-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 34.