http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-032605-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_0bd433e19d43c4d9b2a68ed8443b9a9a |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N43-54 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D239-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-54 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D239-80 |
| filingDate | 2000-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9f70f60d7e57494995947f456668611a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c9adc8b451c09f94f1c6d064a010b842 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_bf55b66f4be28bbba9baa4ec0b5011d6 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3f659f4e54df2c497e7bcfb3928dcfa9 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_da8f286624f1f78196ab0dfd569a91c7 |
| publicationDate | 2003-11-19-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-032605-A1 |
| titleOfInvention | DERIVATIVES (TIONA) AMINOQUINAZOLINONA REPLACED OR SALTS OF THE SAME, INTERMEDIATE COMPOUNDS OF THE SAME, AND PEST CONTROLLERS AND A METHOD FOR USING THEMSELVES |
| abstract | It is known that aminoquinazolinone derivatives are useful as pest controllers in order to find a novel pest controller better, it was found that the compounds derived (thione) aminoquinazolinone and that they have substituents in the phenyl group belonging to the quinazolinone ring, possess the same or better insecticidal effect at a low dosage compared to the known compounds. A substituted (thione) aminoquinazolinone derivative that is represented by the general formula (1), or a salt thereof, wherein R is a hydrogen atom; hydroxyl, formyl, C1-12 alkyl, halo C1-6 alkyl, hydroxy C1-6 alkyl, alkenyl C2-6, C2.6 alkynyl, C1-6 alkoxy, halo C1-6 alkoxy, C1-6 alkoxy C1-3 alkyl , C1-6 alkoxy C1-3 alkoxy C1-3 alkyl, C1-6 alkylthio, C1-6 halo alkyl, C1-6 alkylsulfinyl, C1-6 alkylsulfonyl, C1-6 alkylthio C1-3 alkyl, C1-6 dialkoxy C1 alkyl -3 in which the C1-6 alkoxy groups may be the same or different, unsubstituted amino C1-6 alkyl, substituted C1-6 amino alkyl having one or two substituents that may be the same or different and is selected from the group consisting C1-6 alkyl, halo C1-6 alkyl, C2-6 alkenyl and C2-6 alkynyl, cyano C1-6 alkyl, C1-6 alkylcarbonyl, C1-6 alkoxycarbonyl, C1-3 hydroxycarbonyl C1, C1-6 alkoxycarbonyl C1 -3, unsubstituted aminocarbonyl, substituted aminocarbonyl having one or two substituents that may be the same or different and are selected from the group consisting of C1-6 alkyl, C2-6 alkenyl and C2-6 alkynyl, cyc C 3-6 alkyl C1-3 alkyl, phenyl C1-3 unsubstituted alkyl, phenyl C1-3 substituted alkyl having 1 to 5 substituents on the ring which may be the same or different and are selected from the group consisting of halogen atoms, nitro, cyano, C1-6 alkyl, halo C1-6 alkyl, alkoxy C1-6, halo C1-6 alkoxy, C1-6 alkylthio and halo C1-6 alkylthio, unsubstituted phenylcarbonyl, substituted phenylcarbonyl having ring 1 to 5 substituents that may be the same or different and are selected from the group consisting of halogen, nitro, cyano, C16 alkyl, C1-6 alkyl, C1-6 alkoxy, C1-6 alkoxy halo, C1-6 alkylthio and halo atoms C1-6 alkylthio, unsubstituted phenylthio, substituted phenylthio having 1 to 5 substituents on the ring that may be the same or different and are selected from the group consisting of halogen, nitro, cyano, C1-6 alkyl, C1- halo atoms 6 alkyl, C1-6 alkoxy, C1-6 halo alkoxy, C1-6 alkylthio and C1-6 alkylthio halo, phenylsulfonyl without its stituir, substituted phenylsulfonyl having 1 to 5 substituents on the ring that may be the same or different and is selected from the group consisting of halogen, nitro, cyano, C1-6 alkyl, C1-6 halo halo, C1-6 alkoxy , halo C1-6 alkoxy, alkylthio C1-6 and halo C1-6 alkylthio, phenyl C1-6 alkylsulfonyl, substituted phenyl C1-6 alkylsulfonyl having 1 to 5 substituents on the ring which may be the same or different and are selected from the group consisting of halogen, nitro, cyano, C 1-6 alkyl, C 1-6 alkyl, C 1-6 alkoxy, C 1-6 alkoxy halo, C 1-6 alkylthio and C 1-6 alkyl alkylthio, unsubstituted phenyloxycarbonyl atoms, substituted phenyloxycarbonyl having 1 to 5 substituents on the ring which may be the same or different and is selected from the group consisting of halogen, nitro, cyano, C1-6 alkyl, halo C1-6 alkyl, C1-6 alkoxy, halo C1-6 alkoxy, alkylthio and halo C1-6 alkylthio, unsubstituted phenyloxy alkyl, phenyloxy C1-3 substituted alkyl having 1 to 5 substituents on the ring which may be the same or different and are selected from the group consisting of halogen, nitro, cyano, C1-6 alkyl, halo C1-6 alkyl, C1- alkoxy 6, halo C1-6 alkoxy, alkylthio C1-6 and halo C1-6 alkylthio, phenyl C2-6 alkenyl, substituted phenyl C2-6 alkenyl having 1 to 5 substituents on the ring which may be the same or different and are selected from the group consisting of halogen, nitro, cyano, C1-6 alkyl, halo C1-6 alkyl, C1-6 alkoxy, C1-6 haloxy, C1-6 alkyl, C1-6 alkyl alkylthio and C1- alkylenedioxy atoms 2, phenyl C2-6 unsubstituted alkynyl, phenyl C2-6 substituted alkynyl having 1 to 5 substituents on the ring which may be the same or different and are selected from the group consisting of halogen, nitro, cyano, C1- alkyl atoms 6, halo C1-6 alkyl, C1-6 alkoxy, halo C1-6 alkoxy, C1-6 alkylthio, halo C1-6 alkylthio and C1-2 alkylenedioxy, phenyl C 2-4 C1-3 alkynyl unsubstituted alkyl, C2-4 phenyl C1-3 alkynyl substituted alkyl having 1 to 5 substituents on the ring which may be the same or different and are selected from the group consisting of halogen atoms, nitro, cyano, C1-6 alkyl, halo C1-6 alkyl, alkoxy, halo C1-6 alkoxy, C1-6 alkylthio, halo C1-6 alkylthio and C1-2 alkylenedioxy, 1,3-dioxolan-2-yl C1-3 alkyl , or C1-6 alkyl phthalimido; R1 is a 5- or 6- membered heterocyclic ring that has 1 to 3 heteroatoms that can be the same or different and are selected from the group consisting of the oxygen atom, sulfur atom and nitrogen atom, said heterocyclic ring may have 1 to 5 substituents that may be the same or different and are selected from the group consisting of halogen, cyano, C1-6 alkyl, halo C1-6 alkyl and C1-6 alkoxy groups, and the nitrogen atom in the heterocyclic ring may form an N-oxide group; And it is the atom of an oxygen or a sulfur atom; Z is ûN = C (R2) - (where R2 is a hydrogen atom, C1-6 alkyl or a halo C1-6 alkyl group, or ûN (R3) -CH (R2) - (where R2 is equal to defined above, and R3 is a hydrogen atom, C1-6 alkyl, formyl, C1-3 alkylcarbonyl or C1-3 halocarbonyl; X may be the same or different, and is a bromine atom, an iodine atom, hydroxyl, cyano, C1-6 alkyl, halo C1-10 alkyl, C2-6 alkenyl, halo C2-6 alkenyl, alkynyl C2-6, alkoxy C1-6, halo C1-6 alkoxy, alkylthio C1-6, halo C1-6 alkylthio C 1-6 alkylsulfinyl, C 1-6 alkylsulfinyl, C 1-6 alkylsulfonyl, C 1-6 alkylsulfonyl, C 1-6 halo C 1-6 alkoxyhaloxy, carboxy, C 1-6 alkoxycarbonyl, unsubstituted aminocarbonyl, substituted aminocarbonyl having one or two substituents that may be the same or different and are selected from the group consisting of C1-6 alkyl, C2-6 alkenyl and C2-6 alkynyl, C1-6 carboxy C1-6 alkoxycarbonyl C1-3 alkyl, C1-3 aminocarbonyl alkyl no substitute ir, C1-3 aminocarbonyl substituted alkyl having one or two substituents that may be the same or different and are selected from the group consisting of C1-6 alkyl, C2-6 alkenyl and C2-6 alkynyl sulfonic acid, unsubstituted aminosulfonyl, alkoxysulfonyl C1-6, substituted aminosulfonyl having one or two substituents that may be the same or different and are selected from the group consisting of C1-6 alkyl, C2-6 alkenyl and C2-6 alkynyl, unsubstituted phenyl, substituted phenyl which it possesses in the ring 1 to 5 substituents that may be the same or different and are selected from the group consisting of halogen atom, nitro, cyano, C1-6 alkyl, C1-6 halo alkyl, C1-6 alkoxy, C1-6 alkoxy halo, C1-6 alkylthio, C1-6 halo alkylthio, C1-6 alkoxysulfonyl and substituted aminosulfonyl having one or two substituents that may be the same or different and are selected from the group consisting of C1-6 alkyl, C2-6 alkenyl and C2 alkynyl -6, phenyl C1-3 unsubstituted alkyl, C1-3 phenyl substituted alkyl having 1 to 5 substituents on the ring which may be the same or different and are selected from the group consisting of halogen, nitro, cyano, C1-6 alkyl, C1-6 alkyl halo, C1 alkoxy atoms -6, halo C1-6 alkoxy, C1-6 alkylthio and halo C1-6 alkylthio, unsubstituted phenyloxy, substituted phenyloxy having 1 to 5 substituents on the ring which may be the same or different and are selected from the group consisting of atoms halogen, nitro, cyano, C1-6 alkyl, halo C1-6 alkyl, C1-6 alkoxy, halo C1-6 alkoxy, C1-6 alkylthio and C1-6 alkylthio, unsubstituted pyridyloxy, or substituted pyridyloxy having one or more substituents that may be the same or different and are selected from the group consisting of halogen, nitro, cyano, C1-6 alkyl, halo C1-6 alkyl, C1-6 alkoxy, C1-6 alkoxy halo, C1- alkylthio atoms 6 and halo C1-6 alkylthio, and n is an integer from 0 to 4. A compound useful as an intermediate for the synthetic is of the substituted (thione) aminoquinazolinone derivative, which is represented by formula (2), wherein, X may be the same or different and is a bromine atom, an iodine, hydroxyl, cyano, C1-6 alkyl, halo atom C 1-6 alkyl, C 1-6 alkenyl, C 2-6 alkenyl halo, C 2-6 alkynyl, C 1-6 alkoxy, C 1-6 alkoxy alkoxy, C 1-6 alkylthio, C 1-6 alkylthio halo, C 1-6 alkylsulfinyl, C 1-6 halo -6 alkylsulfinyl, C1-6 alkylsulfonyl, halo C1-6 alkylsulfonyl, halo C1-6 alkoxyhalo C1-6 alkoxy, carboxyl, C1-6 alkoxycarbonyl, unsubstituted aminocarbonyl, substituted aminocarbonyl having one or two substituents which may be the same or different and are selected from the group consisting of C1-6 alkyl, C2-6 alkenyl and C2-6 alkynyl, C1-6 carboxy alkyl, C1-6 alkoxycarbonyl C1-3 alkyl, unsubstituted C1-3 aminocarbonyl, C1-3 aminocarbonyl substituted alkyl having one or two substituents that may be the same or different and are selected from the group consisting of C1 alkyl -6, C2-6 alkenyl and C2-6 alkynyl, sulfonic acid, C1-6 alkoxysulfonyl, sulfonamide possessing a hydrogen atom, C1-6 alkyl, C2-6 alkenyl or C2-6 alkynyl in the nitrogen atom, phenyl unsubstituted, substituted phenyl having 1 to 5 substituents on the ring that may be the same or different and are selected from the group consisting of halogen, nitro, cyano, C1-6 alkyl, halo C1-6 alkyl, C1- alkoxy 6, halo C1-6 alkoxy, alq |
| priorityDate | 1999-11-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 58.