http://rdf.ncbi.nlm.nih.gov/pubchem/patent/AR-012684-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_5c24684033fba97d1ad845ce453a57e3 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P37-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-48 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D333-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D217-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D217-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-448 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D403-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D307-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P1-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P37-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P1-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-34 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-47 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D333-32 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P19-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-472 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D217-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D217-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D307-58 |
| filingDate | 1998-05-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2000-11-08-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | AR-012684-A1 |
| titleOfInvention | ACIDS 6- AND 7-AMINO-TETRAHYDROISOQUINOLINACARBOXILICOS SUBSTITUTED, PROCEDURE FOR ITS PREPARATION, ITS USE IN THE PREPARATION OF A MEDICINAL PRODUCT, MEDICATION THAT CONTAINS THEM AND PROCEDURE FOR ITS PREPARATION |
| abstract | 6- and 7-amino-tetrahydroisoquinolincarboxylic acids substituted, comprising formula (I) and / or a stereoisomeric form of the compound of formula (I) and / or a physiologically compatible salt of the compound of formula (I), representing in it: R1 is: 1. phenyl, 2. phenyl, which is substituted once or twice with: 2.1 C1-6 alkyl, linear, cyclic or branched, 2.2 -OH, 2.3 C1-6-C (O) -O alkyl -, 2.4 C1-6 alkyl-O-, 2.5 C1-6 alkyl-C1-4-alkyl-, 2.6halogen, 2.7 -CF3, 2.8 -CN, 2.9 -NO2, 2.10 HO-C (O) -, 2.11 C1-6alkyl-OC (O) -, 2.12 methylenedioxo, 2.13 R5- (R6) NC (O) -, in which R5 and R6 are the same or different and represent a hydrogen or C1-6 alkyl atom, or 2.14 R5 - (R6) N-, where R5 and R6 are the same or different and represent a hydrogen atom or C1-6 alkyl; 3. a heteroaromatic radical taken from the following group 3.1 to 3.15, which is unsubstituted or substituted as described in 2.1 to 2.14: 3.1 pyrrole, 3.2pyrazole, 3.3 imide zol, 3.4 triazole, 3.5 thiophene, 3.6 thiazole, 3.7 oxazole, 3.8 isoxazole, 3.9 pyridine, 3.10 pyrimidine, 3.11 indole, 3.12 benzothiophene, 3.13 benzimidazole, 3.14 benzoxazole, or 3.15 benzothiazole; 4. -OH and A denoting a bond; 5. -O-R1 4 and A denoting a covalent bond, -CH = CH- or -C ::: C- and wherein R14 denotes 1) C1-6 alkyl, 2) C3-6 cycloalkyl, 3) benzyl or 4) phenyl; 6. -COOH and A denoting a covalent bond, -CH = CH or -C ::: C-; 7. C1-6alkyl; 8. C3-6-cycloalkyl-O-C1-4alkyl; 9. halogen and meaning A covalent bond, -CH = CH- or -C ::: C-, 10. -CN and meaning A covalent bond, -CH = CH- or C ::: C-; 11. -NO2 and A denoting a covalent bond, -CH = CH- or C ::: C-, or 12.-CF3, and R2 representing: 1. HO (H) N- or 2. R7-O-, in that R7 means 2.1 a hydrogen atom, 2.2 C1-6 alkyl, |
| priorityDate | 1997-05-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 74.