title |
Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells/Nrf2 (unknown origin) protein-protein interaction using FITC-LDEETGEFL-NH2 as fluorescent substrate at 0.5 uM preincubated with compound for 30 mins followed by substrate addition and measured after 1 hr by fluorescence polarization assay relative to control |