http://rdf.ncbi.nlm.nih.gov/pubchem/author/MD5_c6f731d716daa23071ddb2d20f79dd15
Outgoing Links
Predicate | Object |
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family-name | Knapp |
name | Stefan Knapp |
given-name | Stefan |
organization-name | Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford Oxford UK Authors' Affiliations: 1Weatherall Institute of Molecular Medicine, University of Oxford, Headington; 2Nuffield Department of Obstetrics and Gynaeoclogy, Women's Centre, John Radcliffe Hospital; 3Nuffield Department of Clinical Medicine, SGC, Oxford, United Kingdom; and 4Xijing Hospital, the Fourth Military Medical University, Shaanxi Province, China Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford, Oxford OX3 7DQ, United Kingdom;; Department of Clinical Pharmacology, University of Oxford, Oxford OX3 7DQ, United Kingdom Nuffield Department of Clinical Medicine, Structural Genomics Consortium, Oxford University, Old Road Campus Research Building, Headington, Oxford OX3 7DQ, U.K. Structural Genomics Consortium, Nuffield Department of Clinical Medicine, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, U.K.; Target Discovery Institute (TDI), University of Oxford, NDM Research Building, Roosevelt Drive, Oxford, OX3 7FZ, U.K. Structural Genomics Consortium (SGC), University of Oxford, Headington, UK; Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Frankfurt, Germany Nuffield Department of Clinical Medicine, Structural Genomics Consortium and Target Discovery Institute, University of Oxford, Oxford OX3 7DQ, United Kingdom Structural Genomics Consortium, Nuffield Department of Clinical Medicine, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, United Kingdom Institute for Pharmaceutical Chemistry, Structural Genomics Consortium, and Buchmann Institute for Molecular Life Sciences, Johann Wolfgang Goethe-University, Frankfurt am Main, Germany. Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences, Goethe University Frankfurt, Frankfurt am Main, Germany Nuffield Department of Clinical Medicine, Structural Genomics Consortium and Target Discovery Institute, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, U.K.; Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University and Buchmann Institute for Molecular Life Sciences, Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany Structural Genomics Consortium, Nuffield Department of Clinical Medicine, University of Oxford, Oxford OX3 7DQ, United Kingdom;; Target Discovery Institute, Nuffield Department of Clinical Medicine, University of Oxford, Oxford OX3 7BN United Kingdom Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Target Discovery Institute, University of Oxford, Oxford OX3 7FZ, U.K.; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences, Goethe University, Max-von Laue Str. 9, 60438 Frankfurt am Main, Germany. Nuffield Department of Clinical Medicine, Target Discovery Institute, University of Oxford, Oxford, 3 7FZ, UK. knapp@pharmchem.uni-frankfurt.de. Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-Universität, Max-von-Laue-Str. 9, 60438, Frankfurt am Main, Germany. knapp@pharmchem.uni-frankfurt.de. 2Aligning Science Across Parkinson's (ASAP) Collaborative Research Network, Chevy Chase, MD 20815, U.S.A.; 3Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences and Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Max-von-Laue-Str. 9, D-60438 Frankfurt am Main, Germany Structural Genomics Consortium, Nuffield Department of Clinical Medicine, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, United Kingdom; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences, Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, United Kingdom; Nuffield Department of Clinical Medicine, Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Oxford OX3 7FZ, United Kingdom Structural Genomics Consortium, Oxford University, Old Road Campus Building, Roosevelt Drive, Oxford, OX3 7DQ, United Kingdom Microbiology and Tumorbiology Center, Karolinska Institutet, 17177 Stockholm, Sweden, Center for Structural Biochemistry, Karolinska Institutet, NOVUM, 14157 Stockholm, Sweden, and Département de Biochimie, Université de Genève, 30 quai E. Ansermet, 1211 Genève 4, Switzerland Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, U.K.; Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Oxford, OX3 7LD, U.K. 2Oxford University, Structural Genomics Consortium, Botnar Research Centre, Oxford, United Kingdom; and Structural Genomics Consortium and Target Discovery Institute, Nuffield Department of Clinical Medicine, University of Oxford, Oxford, United Kingdom *Structural Genomics Consortium, Botnar Research Centre, University of Oxford, Oxford OX3 7LD, United Kingdom; and Structural Genomics Consortium, Oxford University, Old Road Campus Research Building, Old Road Campus, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Target Discovery Institute, Oxford University, NDM Research Building, Old Road Campus, Roosevelt Drive, Oxford OX3 7FZ, U.K. Structural Genomics Consortium, Nuffield Department of Clinical Medicine, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Target Discovery Institute, Nuffield Department of Clinical Medicine, University of Oxford, Roosevelt Drive, Oxford OX3 7BN, U.K.; Institute for Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany Johann Wolfgang Goethe-University Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences 60438 Frankfurt am Main Germany Goethe-University Frankfurt, Institute of Pharmaceutical Chemistry, Frankfurt, Germany. Structural Genomic Consortium (SGC) University of Oxford Oxford OX3 7DQ UK; Target Discovery Institute (TDI) University of Oxford Oxford OX3 7FZ UK; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences Johann Wolfgang Goethe-University 60438 Frankfurt am Main Germany Structural Genomics Consortium, University of Oxford, Old Road Campus Building, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Department of Clinical Pharmacology, University of Oxford, Old Road Campus Building, Roosevelt Drive, Oxford OX3 7DQ, U.K. Structural Genomic Consortium, University of Oxford, Old Road Campus, Oxford OX3 7DQ, United Kingdom; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences, Johann Wolfgang Goethe-University, D-60438, Frankfurt am Main, Germany Target Discovery Institute (TDI), and Structural Genomics Consortium (SGC), University of Oxford, Old Road Campus Research Building, Oxford OX3 7DQ, U.K.; Institute of Pharmaceutical Chemistry and Buchman Institute for Life Sciences, Goethe-University, Max-von-Laue-Strasse 9, 60438 Frankfurt am Main, Germany Structural Genomics Consortium, Buchmann Institute for Life Sciences, Goethe-University Frankfurt, Frankfurt, Germany; Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt, Frankfurt, Germany Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Nuffield Department of Clinical Medicine, Target Discovery Institute (TDI), University of Oxford, Roosevelt Drive, Oxford OX3 7BN, U.K.; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences, Johann Wolfgang Goethe-University, Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany Nuffield Department of Clinical Medicine, SGC, University of Oxford, Oxford OX3 7DQ, U.K.; Nuffield Department of Clinical Medicine, Target Discovery Institute, University of Oxford, Oxford OX3 7FZ, U.K. The Structural Genomic Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Headington, Oxford OX3 7DQ, U.K.; Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Headington, Oxford OX3 7FZ, U.K.; Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Max-von-Laue-Strasse 9 D-60438 Frankfurt am Main, Germany Structural Genomics Consortium, Oxford University, Old Road Campus Research Building, Old Road Campus, Roosevelt Drive, Oxford, OX3 7DQ, U.K.; Department of Clinical Pharmacology, University of Oxford, Old Road Campus Building, Roosevelt Drive, Oxford OX3 7DQ, U.K. Structural Genomics Consortium & Target Discovery Institute University of Oxford, NDMRB Old Road Campus Oxford, OX3 7DQ & OX3 7FZ UK; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences Johann Wolfgang Goethe-University 60438 Frankfurt am Main Germany Institute of Pharmaceutical Chemistry and Buchmann Institute for Life Sciences (BMLS) Goethe University Max-von-Laue-Strasse 9 60438 Frankfurt Germany; Nuffield Department of Clinical Medicine, Structural Genomics Consortium and Target Discovery Institute University of Oxford, Old Road Campus Research Building Roosevelt Drive Oxford OX3 7DQ UK Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences, Frankfurt am Main, Germany; Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Frankfurt am Main, Germany. Electronic address: knapp@pharmchem.uni-frankfurt.de. Nuffield Department of Clinical Medicine, Chemical Genomics Consortium University of Oxford Old Road Campus Research Building, Roosevelt Drive, Headington Oxford OX3 7DQ U.K.; Institute of Pharmaceutical Chemistry and Buchmann Institute for Life Sciences Goethe-University Frankfurt 60438 Frankfurt am Main Germany Structural Genomics Consortium, University of Oxford, OX3 7DQ Oxford, UK. University of Oxford, Structural Genomics Consortium (SGC), Department of Clinical Medicine, Old Road Campus Research Building, Oxford OX3 7DQ, UK ; ;; University of Oxford, Department of Clinical Pharmacology, Old Road Campus Research Building, Oxford OX3 7DQ, UK Target Discovery Institute (TDI) and Structural Genomics Consortium, Oxford University, Oxford, United Kingdom. Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, U.K. Nuffield Department of Clinical Medicine; Structural Genomics Consortium and Target Discovery Institute (TDI) University of Oxford; Oxford OX3 7BN, UK Nuffield Department of Clinical Medicine, Structural Genomics Consortium, Oxford University, Old Road Campus Research Building, Headington, Oxford OX3 7DQ, United Kingdom University of Oxford, Structural Genomics Consortium, Old Road Campus Research Centre, Oxford OX3 7DQ, England, UK 3 Structural Genomics Consortium, Buchmann Institute for Life Sciences, Goethe University Frankfurt Frankfurt Germany; Institute of Pharmaceutical Chemistry, Goethe University Frankfurt Frankfurt Germany; German Cancer Network (DKTK) Frankfurt Germany Nuffield Department of Clinical Medicine, Old Road Campus Research Building, University of Oxford, Oxford OX3 7BN, UK Nuffield Department of Clinical Medicine, Structural Genomics Consortium, Oxford, UK.; Nuffield Department of Clinical Medicine, Target Discovery Institute, Oxford, UK. Nuffield Department of Clinical Medicine, Structural Genomics Consortium and Target Discovery Institute (TDI), University of Oxford, Oxford, United Kingdom Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, United Kingdom; Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Oxford OX3 7LD, United Kingdom SGC, University of Oxford, Oxford OX3 7DQ, United Kingdom Department of Chemistry, Pharmacia, Viale Pasteur 10, 20014 Nerviano (MI), Italy Buchmann Institute for Molecular Life Sciences, Structural Genomics Consortium, Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany; Institute for Pharmaceutical Chemistry, Max von Lauestrasse 9, Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany; Translational cancer network DKTK site Frankfurt/Mainz and Frankfurt Cancer Institute (FCI), Johann Wolfgang Goethe-University, D-60438 Frankfurt am Main, Germany Discovery Research Oncology, Department of Chemistry, Pharmacia Corporation, Viale Pasteur 10, 20014 Nerviano, Italy, San Raffaele Scientific Institute, via Olgettina 58, 20132 Milano, Italy, Bioindustry Park del Canavese Spa, Via Ribes 5, 10010 Colleretto Giacosa, Italy, San Raffaele University, via Olgettina 58, 20132 Milano, Italy, and Dulbecco Telethon Institute, c/o San Raffaele Scientific Institute, Via Olgettina 58, 20132 Milano, Italy Nuffield Department of Clinical Medicine Oxford UK; Department of Clinical PharmacologyOxford University Oxford UK Structural Genomics Consortium, University of Oxford, Oxford OX3 7LD, United Kingdom; Institute of Pharmaceutical Chemistry Buchmann Institute for Molecular Life Sciences Goethe University Frankfurt/Main Germany Target Discovery Institute (TDI), Nuffield Department of Medicine, University of Oxford, Oxford, OX37FZ, United Kingdom; Institute for Pharmaceutical Chemistry and Buchmann Institute for Molecular Life Sciences (BMLS), Johann Wolfgang Goethe University, Frankfurt am Main, 60438, Germany Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Target Discovery Institute, Nuffield Department of Medicine, University of Oxford, Roosevelt Drive, Oxford OX3 7FZ, U.K. Nuffield Department of Medicine, Structural Genomics Consortium, Old Road Campus Research Building, Oxford University, Oxford, OX3 7DQ, United Kingdom; Institute of Pharmaceutical Chemistry and Buchmann Institute for Life Sciences (BMLS), Structure Genomics Consortium, Goethe-University Frankfurt, Max von Lauestrasse 9, 60438 Frankfurt am Main, Germany Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt, 60438 Frankfurt, Germany; Structural Genomics Consortium, BMLS, Goethe-University Frankfurt, 60438 Frankfurt, Germany Nuffield Department of Clinical Medicine, University of Oxford, Structural Genomics Consortium, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences, Johann Wolfgang Goethe-University, Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Oxford, OX3 7FZ, United Kingdom; Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, United Kingdom; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences (BMLS), Johann Wolfgang Goethe University, Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Oxford OX3 7DQ, United Kingdom;; Institute for Pharmaceutical Chemistry, Goethe University Frankfurt, 60438 Frankfurt, Germany;; Buchmann Institute for Life Sciences, Goethe University Frankfurt, 60438 Frankfurt, Germany; 1 Structural Genomics Consortium, University of Oxford, Headington, Oxford OX37DQ, UK, 2Structural Genomics Consortium, University of Toronto, Toronto, ON M5G1L7, Canada, 3Oxford NIHR Biomedical Research Unit, Botnar Research Centre, 4Nuffield Department of Clinical Medicine, Old Road Campus, University of Oxford, Headington, Oxford, OX3 7DQ, UK and 5Department of Pharmacology and Toxicology, University of Toronto, ON M5S1A8, Canada The Structural Genomic Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Headington, Oxford OX3 7DQ, U.K.; Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Headington, Oxford OX3 7FZ, U.K. Institute for Pharmaceutical Chemistry Structural Genomics Consortium Johann Wolfgang Goethe-University Max-von-Laue-Strasse 15 60438 Frankfurt am Main Germany Structural Genomics Consortium, University of Oxford, Botnar Research Centre, Oxford OX3 7LD, U.K. Philipps-Universität Marburg, Institut für Molekularbiologie und Tumorforschung, 35037 Marburg, Germany DIBIT, San Raffaele Scientific Institute, via Olgettina 58, 2032 Milano, Italy, and Pharmacia & Upjohn, Discovery Research Oncology, Department of Structural Chemistry, Viale Pasteur 10, 20014 Nerviano, Italy Target Discovery Institute and Structural Genomics Consortium, Oxford University, Oxford, UK. knapp@pharmchem.uni-frankfurt.de. Goethe-University Frankfurt, Institute of Pharmaceutical Chemistry and Buchmann Institute for Life Sciences, Frankfurt am Main, Germany. knapp@pharmchem.uni-frankfurt.de. German Cancer Network (DKTK), Frankfurt am Main, Germany. knapp@pharmchem.uni-frankfurt.de. Structural Genomics Consortium (SGC) & Target Discovery Institute Nuffield Department of Medicine University of Oxford, NDM Research Building Roosevelt Drive Oxford OX3 7FZ UK; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences Johann Wolfgang Goethe University 60438 Frankfurt am Main Germany Institute of Pharmaceutical Chemistry, Goethe-University Frankfurt, 60438 Frankfurt, Germany; Structural Genomics Consortium (SGC), Buchmann Institute for Life Sciences, Goethe-University Frankfurt, 60438 Frankfurt, Germany; German Cancer Network (DKTK), Frankfurt/Mainz, 60438 Frankfurt, Germany Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, United Kingdom; Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Oxford, OX3 7FZ, United Kingdom; Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Max-von-Laue-Str. 9, D-60438 Frankfurt am Main, Germany Authors' Affiliations: Departments of 1Neurological Surgery and 2Cancer Biology, Vanderbilt University Medical Center, Nashville, Tennessee; Departments of 3Oncology and 4Geriatrics, the Second Affiliated Hospital, 5Department of Oncology, the First Affiliated Hospital, Nanjing Medical University, Nanjing, China; and 6Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Oxford, United Kingdom Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 3TA, U.K. Authors' Affiliations: 1Structural Genomics Consortium and 2Target Discovery Institute, Nuffield Department of Clinical Medicine, University of Oxford, Oxford; 3School of Cancer Sciences, University of Birmingham; 4Department of Cellular Pathology, Queen Elizabeth Medical Centre, Birmingham; 5Pfizer Worldwide Medicinal Chemistry, Pfizer Worldwide R&D, Ramsgate Road, Sandwich, United Kingdom; 6Laboratory for Childhood Leukemia, Department of Biomedicine, University of Basel and Basel University Children's Hospital, Basel, Switzerland; 7Department of Biochemistry and Molecular Biology, School of Medicine and Health Sciences, George Washington University, Washington, DC; 8Department of Medical Oncology, Dana-Farber Cancer Institute; and 9Department of Medicine, Harvard Medical School, Boston, Massachusetts; Authors' Affiliations: 1Structural Genomics Consortium and 2Target Discovery Institute, Nuffield Department of Clinical Medicine, University of Oxford, Oxford; 3School of Cancer Sciences, University of Birmingham; 4Department of Cellular Pathology, Queen Elizabeth Medical Centre, Birmingham; 5Pfizer Worldwide Medicinal Chemistry, Pfizer Worldwide R&D, Ramsgate Road, Sandwich, United Kingdom; 6Laboratory for Childhood Leukemia, Department of Biomedicine, University of Basel and Basel University Children's Hospital, Basel, Switzerland; 7Department of Biochemistry and Molecular Biology, School of Medicine and Health Sciences, George Washington University, Washington, DC; 8Department of Medical Oncology, Dana-Farber Cancer Institute; and 9Department of Medicine, Harvard Medical School, Boston, Massachusetts; Authors' Affiliations: 1Structural Genomics Consortium and 2Target Discovery Institute, Nuffield Department of Clinical Medicine, University of Oxford, Oxford; 3School of Cancer Sciences, University of Birmingham; 4Department of Cellular Pathology, Queen Elizabeth Medical Centre, Birmingham; 5Pfizer Worldwide Medicinal Chemistry, Pfizer Worldwide R&D, Ramsgate Road, Sandwich, United Kingdom; 6Laboratory for Childhood Leukemia, Department of Biomedicine, University of Basel and Basel University Children's Hospital, Basel, Switzerland; 7Department of Biochemistry and Molecular Biology, School of Medicine and Health Sciences, George Washington University, Washington, DC; 8Department of Medical Oncology, Dana-Farber Cancer Institute; and 9Department of Medicine, Harvard Medical School, Boston, Massachusetts Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, United Kingdom Nuffield Department of Clinical Medicine, Structural Genomics Consortium, Oxford University, Old Road Campus Research Building, Headington, Oxford OX3 7DQ, United Kingdom; Nuffield Department of Clinical Medicine, Target Discovery Institute, Oxford University, NDM Research Building, Oxford OX3 7FZ, United Kingdom Institute of Pharmaceutical Chemistry, Goethe University Frankfurt, Frankfurt 60438, Germany; Structural Genomics Consortium, BMLS, Goethe University Frankfurt, Frankfurt 60438, Germany Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe University, Frankfurt am Main, Germany; Structure Genomics Consortium, Johann Wolfgang Goethe University, Buchmann Institute for Molecular Life Sciences, Frankfurt am Main, Germany Department of Biochemistry, Chemistry and Pharmacy, Institute for Pharmaceutical Chemistry Goethe University Frankfurt Germany; Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences Goethe University Frankfurt Germany Nuffield Department of Clinical Medicine, Target Discovery Institute (TDI) and Structural Genomics Consortium (SGC) University of Oxford Oxford UK Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford, Oxford OX3 7DQ, England, UK 3 Institute of Pharmaceutical Chemistry Goethe University Frankfurt am Main Germany Institute of Pharmaceutical Chemistry Goethe University Frankfurt Germany; Structural Genomics Consortium Buchmann Institute for Molecular Life Sciences (BMLS) Goethe University Frankfurt Germany Nuffield Department of Clinical Medicine, University of Oxford, Structural Genomics Consortium, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, UK; Nuffield Department of Clinical Medicine, University of Oxford, Target Discovery Institute, Roosevelt Drive, Oxford, OX3 7FZ, UK Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Headington, Oxford OX3 7DQ, U.K. Institute for Pharmaceutical Chemistry and Buchmann Institute for Molecular Life Sciences (S.K.), Goethe University, Frankfurt am Main, Germany. 1Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Oxford, United Kingdom.; 3Nuffield Department of Clinical Medicine, Target Discovery Institute (TDI), University of Oxford, Oxford, United Kingdom. Institute of Pharmaceutical Chemistry, Johann Wolfgang Goethe University, Max-von-Laue-Str. 9, 60438Frankfurt am Main, Germany; Buchmann Institute for Molecular Life Sciences and Structural Genomics Consortium (SGC), Max-von-Laue-Str. 15, 60438Frankfurt am Main, Germany; Frankfurt Cancer Institute, Goethe University, Frankfurt am Main60596, Germany Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Oxford OX3 7DQ, UK. Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Headington, Oxford OX3 7DQ, United Kingdom; Nuffield Department of Clinical Medicine, Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Headington, Oxford OX3 7FZ, United Kingdom; Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Max-von-Laue-Str. 9, D-60438 Frankfurt am Main, Germany Structural Genomics Consortium, Institute for Pharmaceutical Chemistry and Buchmann Institute for Molecular Life Sciences, Johann Wolfgang Goethe-University, Max-von-Laue-Str. 9, D-60438 Frankfurt am Main, Germany University of Oxford, Nuffield Department of Clinical Medicine, Structural Genomics Consortium, Old Road Campus Research Building, Roosevelt Drive, Headington, Oxford OX3 7DQ, U.K. The Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford, Headington, Oxford OX3 7DQ, UK; Target Discovery Institute, Nuffield Department of Medicine, University of Oxford, Headington, Oxford OX3 7FZ, UK; Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Sciences, Frankfurt am Main D-60438, Germany Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, United Kingdom; Target Discovery Institute, Nuffield Department of Clinical Medicine, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, United Kingdom Fachbereich Biochemie, Chemie und Pharmazie Institut für Pharmazeutische Chemie, Goethe‐University Frankfurt Frankfurt Am Main Germany 7Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Oxford, United Kingdom. The Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Headington, Oxford OX3 7DQ, U.K.; Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Headington, Oxford OX3 7FZ, U.K.; Department of Pharmaceutical Chemistry and Buchmann Institute for Life Sciences, Goethe University Frankfurt, 60438 Frankfurt am Main, Germany Structural Genomics Consortium, Nuffield Department of Clinical Medicine, University of Oxford, Oxford OX3 7DQ, United Kingdom;; Target Discovery Institute, Nuffield Department of Clinical Medicine, University of Oxford, Oxford OX3 7FZ, United Kingdom;; Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, 60438 Frankfurt am Main, Germany Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, United Kingdom Structural Genomics Consortium; Nuffield Department of Clinical Medicine; University of Oxford; Oxford OX3 7DQ; UK Nuffield Department of Medicine, Structural Genomics Consortium, University of Oxford, Oxford, United Kingdom; Institute for Pharmaceutical Chemistry, Goethe University, Frankfurt, Germany; Buchmann Institute for Molecular Life Science, Goethe University, Frankfurt, Germany University of Oxford, Target Discovery Institute (TDI) and Structural Genomics Consortium (SGC), Old Road Campus Research Building, Oxford OX3 7DQ, U.K. Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Buchmann Institute for Molecular Life Sciences, Max-von-Laue-Strasse 15, D-60438 Frankfurt am Main, Germany; Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Max-von-Laue-Strasse 9, D-60438 Frankfurt am Main, Germany Biology and Chemistry Departments, Nerviano Medical Sciences, Viale Pasteur 10, 20014 Nerviano (Milan), Italy Contribution from the Chemistry Department and Biology Department, Pharmacia, Viale Pasteur 10, 20014 Nerviano (MI), Milano, Italy, and Structural, Analytical & Medicinal Chemistry Department, Pharmacia, 301 Henrietta Street, Kalamazoo, Michigan 49001 Structural Genomics Consortium (SGC), Botnar Research Centre, Oxford University, Oxford OX3 7LD, U.K., and School of Chemistry, University of Leeds, Leeds, LS2 9JT, U.K. Department of Pharmaceutical Chemistry, University of Frankfurt, Frankfurt, Germany Authors' Affiliations: 1Institut Albert Bonniot, CRI INSERM/UJF U823, Team 3 “Polarity, Development and Cancer”, Rond-point de la Chantourne, La Tronche Cedex; 2CEA, DSV, iRTSV/CMBA; 3INSERM, U1036, CEA, iRTSV/BCI, Grenoble; 4Institut Curie, Centre de Recherche; 5CNRS, UMR 176, Paris; 6Institut Curie, Centre de Recherche, Bâtiment 112, Université Paris-Sud, Orsay; 7INSERM UMR 911, Centre de Recherche en Oncologie biologique et Oncopharmacologie, Aix-Marseille Université, Marseille; 8Centre Commun de Quantimétrie, Faculté de Médecine Rockefeller; 9Equipe Labellisée Ligue 2009, Institut de Biologie et Chimie des Protéines FR 3302, BM2SI UMR 5086 CNRS/Université Lyon 1; 10INSERM 590, Faculté Rockefeller, Lyon, France and Université Lyon 1, ISPB, Lyon, France; 11St Vincent's Institute of Medical Research; 12The University of Melbourne, Department of Medicine, St Vincent's Hospital, Fitzroy, Victoria, Australia; and 13Department of Clinical Pharmacology, Oxford University, Oxford, United Kingdom Target Discovery Institute (TDI), and Structural Genomics Consortium (SGC), University of Oxford, Old Road Campus Research Building, Oxford OX3 7DQ, United Kingdom Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford, Headington, OX3 7DQ Oxford, United Kingdom; Target Discovery Institute, University of Oxford, NDM Research Building, Roosevelt Drive, Oxford OX3 7FZ, U.K.; Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Goethe-University, Institute for Pharmaceutical Chemistry and Buchmann Institute for Life Science, Campus Riedberg, Max-von Laue Str. 9, 60438 Frankfurt am Main, Germany University of Oxford, Nuffield Department of Clinical Medicine, Structural Genomics Consortium, Old Road Campus Research Building, Oxford OX3 7DQ, United Kingdom Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, U.K. Institute for Pharmaceutical Chemistry, Structural Genomics Consortium, Johann Wolfgang Goethe-University, Frankfurt am Main, Germany. knapp@pharmchem.uni-frankfurt.de. Frankfurt Cancer Institute (FCI), Frankfurt am Main, Germany; Goethe University Frankfurt, Department of Biochemistry, Chemistry and Pharmacy, Institute for Pharmaceutical Chemistry, Frankfurt am Main, Germany Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Oxford, UK 5 Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Old Road Campus, Roosevelt Drive, Oxford OX3 7DQ, U.K.; Target Discovery Institute, University of Oxford, NDM Research Building, Old Road Campus, Roosevelt Drive, Oxford OX3 7FZ, U.K. |
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Total number of triples: 472.